SCHEMBL18898692

SCHEMBL18898692

CCC(C)n1ncc2cnc(C(C)C)nc21

nearest known ligand 0.30

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.30
CDK1 P06493 1/20 0.30
AURKB Q96GD4 1/20 0.30
CDK4 P11802 1/20 0.30
CCND1 P24385 1/20 0.30
CCND2 P30279 1/20 0.30
CCND3 P30281 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
ADORA3 P0DMS8 1/20 0.30
ADORA2A P29274 1/20 0.30
ADORA2B P29275 1/20 0.30
ADORA1 P30542 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17807781 0.83 AURKA (0.40) AURKACDK1AURKBADORA3ADORA2A
SCHEMBL18898669 0.77 XDH (0.36) CDK4CCND1CCND2CCND3
SCHEMBL19421539 0.74 PI4KA (0.34) AURKACDK1AURKBADORA2AADORA1
SCHEMBL19200217 0.73
SCHEMBL29311529 0.71 KDM4E (0.45) CDK4CCND1CCND2CCND3L3MBTL1
SCHEMBL31469698 0.71 KMO (0.39) CDK4CCND1CCND2CCND3L3MBTL1
SCHEMBL25164705 0.70 HTR2A (0.38)
SCHEMBL15970721 0.70 HDAC8 (0.46) ADORA3ADORA2AADORA2BADORA1
SCHEMBL25164210 0.69 CYP17A1 (0.38)
SCHEMBL25164208 0.68 RIPK1 (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9663520-B2 Bicyclic bromodomain inhibitors ZENITH EPIGENETICS LTD. (CA) 2017-05-30 US disclosed