SCHEMBL18924452

SCHEMBL18924452

CN(C)C(=O)c1ccc(-c2ccc3[nH]c(=O)[nH]c3c2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIK1 P39086 2/20 0.54
GRIK2 Q13002 1/20 0.54
GRIK3 Q13003 1/20 0.54
PDE3B Q13370 1/20 0.53
PDE3A Q14432 1/20 0.53
ERN1 O75460 3/20 0.49
GRIA1 P42261 5/20 0.46
CACNG8 Q8WXS5 4/20 0.46
NCOA1 Q15788 1/20 0.46
NCOA3 Q9Y6Q9 1/20 0.46
MMP2 P08253 1/20 0.46
MMP9 P14780 1/20 0.46
MMP8 P22894 1/20 0.46
LMNA P02545 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
CLK4 Q9HAZ1 1/20 0.44
MAPT P10636 2/20 0.43
LRRK2 Q5S007 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6766299 0.87 MEN1 (0.46) GRIK1GRIK2GRIK3GRIA1CACNG8
SCHEMBL10626283 0.77 ALDH1A1 (0.64) ERN1NCOA1NCOA3MMP2MMP9
SCHEMBL22220936 0.74 PTGS2 (0.56) ERN1CYP1A2CYP3A4MAPTLRRK2
SCHEMBL20838850 0.74 GRIA1 (0.49) GRIK1PDE3BPDE3AGRIA1CACNG8
SCHEMBL18632516 0.72 PDE3B (0.67) GRIK1GRIK2GRIK3PDE3BPDE3A
SCHEMBL22259504 0.72 CYP3A4 (0.50) ERN1MMP2MMP9MMP8LMNA
SCHEMBL22259503 0.72 GSK3B (0.56) ERN1CLK4LRRK2MAPK1
SCHEMBL2455635 0.72 CLK4 (0.53) ERN1LMNACYP1A2CYP3A4CYP2C9
SCHEMBL1119917 0.71 MAPT (0.57) LMNAMAPTALDH1A1KDM4EMAPK1
SCHEMBL1004649 0.71 ALDH1A1 (0.73) ERN1NCOA1NCOA3MMP2MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9670142-B2 1,3-diaminocyclopentane carboxamide derivatives MERCK PATENT GMBH (DE) 2017-06-06 US disclosed