SCHEMBL18933602

SCHEMBL18933602

COCc1cccc(N2CC(OC)C2)c1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AGXT P21549 3/20 0.46
MIF P14174 1/20 0.40
OPRM1 P35372 2/20 0.39
GHSR Q92847 1/20 0.39
PRMT6 Q96LA8 1/20 0.38
OPRD1 P41143 1/20 0.36
OPRK1 P41145 1/20 0.36
MAPT P10636 1/20 0.35
TSHR P16473 1/20 0.35
CACNA2D1 P54289 3/20 0.34
SLC6A2 P23975 2/20 0.34
JAK1 P23458 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19251341 0.79 AGXT (0.71) AGXTPRMT6MAPTTSHRCACNA2D1
SCHEMBL38660066 0.77 NPY1R (0.43) MAPT
SCHEMBL21256823 0.77 ADRB1 (0.50) MAPT
SCHEMBL38660314 0.77 ADRB1 (0.56) MAPTTSHR
SCHEMBL18920849 0.76 AOC2 (0.44) MAPT
SCHEMBL13451177 0.75 ADRB1 (0.62) AGXT
SCHEMBL14288609 0.75 AGXT (0.73) AGXTPRMT6
SCHEMBL31511085 0.74 BPTF (0.48) MAPT
SCHEMBL28994927 0.72 ALDH1A1 (0.41) MAPTTSHR
SCHEMBL30286639 0.72 ALDH1A1 (0.41) MAPTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017093299-A1 1,3,4-THIADIAZOLE COMPOUNDS AND THEIR USE IN TREATING CANCER ASTRAZENECA AB (SE) 2017-06-08 WO disclosed