SCHEMBL18940403

SCHEMBL18940403

C=Cc1ccc(C(=O)Nc2cn(Cc3cc(F)c(F)c(F)c3)cn2)nn1

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 10/20 0.37
CDK5 Q00535 1/20 0.36
CDK5R1 Q15078 1/20 0.36
MAP3K5 Q99683 1/20 0.36
SCD O00767 1/20 0.35
P2RY14 Q15391 1/20 0.33
P2RX7 Q99572 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18940396 0.85 JUN (0.40) RIPK1CDK5CDK5R1MAP3K5SCD
SCHEMBL20083627 0.85 RIPK1 (0.42) RIPK1CDK5CDK5R1MAP3K5SCD
SCHEMBL19645076 0.84 TAS2R8 (0.37) RIPK1CDK5CDK5R1P2RY14
SCHEMBL18940399 0.84 MAP3K5 (0.39) RIPK1CDK5CDK5R1MAP3K5SCD
SCHEMBL18961333 0.78 MAPK7 (0.35) RIPK1CDK5CDK5R1MAP3K5P2RY14
SCHEMBL18961351 0.74 RIPK1 (0.34) RIPK1CDK5CDK5R1MAP3K5P2RY14
SCHEMBL18940435 0.74 TAS2R8 (0.36) RIPK1CDK5CDK5R1MAP3K5P2RY14
SCHEMBL21533354 0.74 RIPK1 (0.44) RIPK1CDK5CDK5R1MAP3K5P2RY14
SCHEMBL18961374 0.73 MAP3K5 (0.41) RIPK1CDK5CDK5R1MAP3K5SCD
SCHEMBL18961316 0.72 KMT2A (0.45) RIPK1CDK5CDK5R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11661397-B2 1,4-disubstituted imidazole derivative Sumitomo Pharma Co., Ltd. (JP) 2023-05-30 US disclosed
US-11661397-B2 1,4-disubstituted imidazole derivative Sumitomo Pharma Co., Ltd. (JP) 2023-05-30 US disclosed
US-11661397-B2 1,4-disubstituted imidazole derivative Sumitomo Pharma Co., Ltd. (JP) 2023-05-30 US disclosed
US-20210171440-A1 1,4-DISUBSTITUTED IMIDAZOLE DERIVATIVE Sumitomo Pharma Co., Ltd. (JP) 2021-06-10 US disclosed
US-20210171440-A1 1,4-DISUBSTITUTED IMIDAZOLE DERIVATIVE Sumitomo Pharma Co., Ltd. (JP) 2021-06-10 US disclosed
CN-107922386-B 1, 4-disubstituted imidazole derivatives 大日本住友制药株式会社 2021-04-02 CN disclosed
US-10807945-B2 1,4-disubstituted imidazole derivative SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) 2020-10-20 US disclosed
US-10807945-B2 1,4-disubstituted imidazole derivative SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) 2020-10-20 US disclosed
EP-3312170-A1 1,4-DI-SUBSTITUTED IMIDAZOLE DERIVATIVE Sumitomo Dainippon Pharma Co., Ltd. (JP) 2018-04-25 EP disclosed
US-9828362-B2 1,4-disubstituted imidazole derivative SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) 2017-11-28 US disclosed
US-20170166552-A1 1,4-DISUBSTITUTED IMIDAZOLE DERIVATIVE Sumitomo Pharma Co., Ltd. (JP) 2017-06-15 US disclosed
US-20170166552-A1 1,4-DISUBSTITUTED IMIDAZOLE DERIVATIVE Sumitomo Pharma Co., Ltd. (JP) 2017-06-15 US disclosed
US-20170166552-A1 1,4-DISUBSTITUTED IMIDAZOLE DERIVATIVE Sumitomo Pharma Co., Ltd. (JP) 2017-06-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170166552-A1 1,4-DISUBSTITUTED IMIDAZOLE DERIVATIVE NR4A3, NR0B1, NR2C2 RIPK1 3318/4885CDK5 1398/4885CDK5R1 936/4885
US-20210171440-A1 1,4-DISUBSTITUTED IMIDAZOLE DERIVATIVE NR4A3, NR0B1, NR2C2 RIPK1 3318/4885CDK5 1398/4885CDK5R1 936/4885
US-11661397-B2 1,4-disubstituted imidazole derivative NR4A3, NR0B1, NR2C2 RIPK1 3318/4885CDK5 1398/4885CDK5R1 936/4885
US-10807945-B2 1,4-disubstituted imidazole derivative NR0B1, NR4A3, H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16 RIPK1 2366/4885CDK5 1246/4885CDK5R1 916/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.