SCHEMBL1894375

SCHEMBL1894375

Cc1cn([C@@H]2O[C@H](COP(=O)(O)NC(=O)[C@@H](N)Cc3c[nH]cn3)[C@@H](O)[C@H]2O)c(=O)[nH]c1=O

nearest known ligand 0.55

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DNPH1 O43598 1/20 0.45
DTYMK P23919 2/20 0.44
P2RY6 Q15077 11/20 0.43
P2RY14 Q15391 4/20 0.43
NT5E P21589 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1894008 0.91 DNPH1 (0.44) DNPH1DTYMKP2RY6P2RY14NT5E
SCHEMBL1895916 0.87 P2RY6 (0.55) P2RY6P2RY14
SCHEMBL1891822 0.84 DNPH1 (0.50) DNPH1P2RY6P2RY14NT5E
SCHEMBL1891030 0.81 P2RY2 (0.52)
SCHEMBL1890617 0.81 TGM2 (0.63) NT5E
SCHEMBL1889579 0.79 P2RY1 (0.61) DNPH1NT5E
SCHEMBL1893832 0.78 P2RY6 (0.53) P2RY6P2RY14
SCHEMBL1886156 0.78 DNPH1 (0.49) DNPH1P2RY6P2RY14NT5E
Histidine SCHEMBL1895268 0.77 P2RY6 (0.54) P2RY6P2RY14
SCHEMBL1892466 0.75 DUT (0.59) P2RY6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8242087-B2 Phosphate modified nucleosides useful as substrates for polymerases and as antiviral agents K.U.LEUVEN RESEARCH & DEVELOPMENT (BE) 2012-08-14 US claimed
US-20110112046-A9 PHOSPHATE MODIFIED NUCLEOSIDES USEFUL AS SUBSTRATES FOR POLYMERASES AND AS ANTIVIRAL AGENTS K.U. LEUVEN RESEARCH & DEVELOPMENT (BE) 2011-05-12 US claimed
US-20100093656-A1 PHOSPHATE MODIFIED NUCLEOSIDES USEFUL AS SUBSTRATES FOR POLYMERASES AND AS ANTIVIRAL AGENTS K.U. LEUVEN RESEARCH & DEVELOPMENT (BE) 2010-04-15 US claimed
EP-2144921-A2 PHOSPHATE MODIFIED NUCLEOSIDES USEFUL AS SUBSTRATES FOR POLYMERASES AND AS ANTIVIRAL AGENTS K.U. Leuven Research and Development (BE) 2010-01-20 EP claimed
WO-2008104408-A2 PHOSPHATE MODIFIED NUCLEOSIDES USEFUL AS SUBSTRATES FOR POLYMERASES AND AS ANTIVIRAL AGENTS K. U. LEUVEN RESEARCH & DEVELOPMENT (BE) 2008-09-04 WO claimed
US-8242087-B2 Phosphate modified nucleosides useful as substrates for polymerases and as antiviral agents K.U.LEUVEN RESEARCH & DEVELOPMENT (BE) 2012-08-14 US disclosed
US-20110112046-A9 PHOSPHATE MODIFIED NUCLEOSIDES USEFUL AS SUBSTRATES FOR POLYMERASES AND AS ANTIVIRAL AGENTS K.U. LEUVEN RESEARCH & DEVELOPMENT (BE) 2011-05-12 US disclosed
US-20100093656-A1 PHOSPHATE MODIFIED NUCLEOSIDES USEFUL AS SUBSTRATES FOR POLYMERASES AND AS ANTIVIRAL AGENTS K.U. LEUVEN RESEARCH & DEVELOPMENT (BE) 2010-04-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110112046-A9 PHOSPHATE MODIFIED NUCLEOSIDES USEFUL AS SUBSTRATES FOR POLYMERASES AND AS ANTIVIRAL AGENTS MTAP, POLRMT, PNP DNPH1 473/4885DTYMK 79/4885P2RY6 590/4885
US-20100093656-A1 PHOSPHATE MODIFIED NUCLEOSIDES USEFUL AS SUBSTRATES FOR POLYMERASES AND AS ANTIVIRAL AGENTS MTAP, POLRMT, PNP DNPH1 473/4885DTYMK 79/4885P2RY6 590/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.