SCHEMBL1894474

SCHEMBL1894474

COc1cc2nccc(Oc3ccc(N(C(=O)O)c4ccccc4)cc3)c2cc1C#N

nearest known ligand 0.56

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AXL P30530 3/20 0.56
MET P08581 2/20 0.56
PDGFRA P16234 11/20 0.53
KDR P35968 7/20 0.53
KIT P10721 2/20 0.51
FGFR2 P21802 3/20 0.50
PDGFRB P09619 2/20 0.50
CSF1R P07333 1/20 0.50
FLT4 P35916 1/20 0.50
FLT3 P36888 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5826134 0.89 PDGFRA (0.66) AXLPDGFRAKDRKITFGFR2
SCHEMBL5825299 0.86 PDGFRA (0.53) AXLMETPDGFRAKDRKIT
SCHEMBL5825967 0.84 FGFR2 (0.68) AXLPDGFRAKDRKITFGFR2
SCHEMBL1893941 0.82 PDGFRA (0.79) AXLMETPDGFRAKDRKIT
SCHEMBL5825195 0.82 PDGFRA (0.62) PDGFRAKDRKITFGFR2PDGFRB
SCHEMBL2174773 0.81 MET (0.61) AXLMETPDGFRAKDRKIT
SCHEMBL5825989 0.81 PDGFRA (0.61) AXLMETPDGFRAKDRKIT
SCHEMBL14967576 0.81 MET (0.60) AXLMETPDGFRAKDRKIT
SCHEMBL1893637 0.80 PDGFRA (0.80) AXLMETPDGFRAKDRKIT
SCHEMBL5825677 0.80 PDGFRA (0.60) AXLMETPDGFRAKDRKIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8372981-B2 Nitrogen-containing aromatic derivatives EISAI R&D MANAGEMENT CO., LTD. (JP) 2013-02-12 US disclosed
US-20110118470-A1 NITROGEN-CONTAINING AROMATIC DERIVATIVES FUNAHASHI YASUHIRO 2011-05-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110118470-A1 NITROGEN-CONTAINING AROMATIC DERIVATIVES GNG2, GCG, FRG1 AXL 3184/4885MET 1619/4885PDGFRA 3135/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.