SCHEMBL18960386

SCHEMBL18960386

Cc1nc(Oc2ccccc2)ccc1I

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 1/20 0.44
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
MAPT P10636 3/20 0.44
MAPK1 P28482 3/20 0.44
HPGD P15428 2/20 0.44
CYP1A2 P05177 2/20 0.44
CYP2C9 P11712 2/20 0.44
CYP2C19 P33261 2/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
ATM Q13315 1/20 0.44
HTT P42858 3/20 0.42
LMNA P02545 1/20 0.42
BCAT2 O15382 1/20 0.42
ALDH1A1 P00352 2/20 0.41
EGLN1 Q9GZT9 1/20 0.40
KDM4E B2RXH2 1/20 0.40
HSD17B10 Q99714 1/20 0.40
TSHR P16473 2/20 0.39
LTA4H P09960 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18960378 0.81 MEN1 (0.46) MAP4K4MEN1KMT2AMAPTMAPK1
SCHEMBL18957388 0.78 BCAT2 (0.50) MAP4K4MEN1KMT2AMAPTMAPK1
SCHEMBL28245881 0.78 MEN1 (0.44) MAP4K4MEN1KMT2AMAPTMAPK1
SCHEMBL11169364 0.78 MAPT (0.49) MAP4K4MEN1KMT2AMAPTMAPK1
SCHEMBL26137908 0.78 KMT2A (0.44) MAP4K4MEN1KMT2AMAPTMAPK1
SCHEMBL19421238 0.75 MAPT (0.41) MAP4K4MEN1KMT2AMAPTMAPK1
SCHEMBL18774086 0.74 NNMT (0.48) KMT2ACYP1A2HTTALDH1A1TDP1
SCHEMBL16511924 0.74 MAP4K4 (0.54) MAP4K4MEN1KMT2AMAPTMAPK1
SCHEMBL5526629 0.74 MEN1 (0.41) MAP4K4MEN1KMT2AMAPTMAPK1
SCHEMBL16805396 0.74 L3MBTL1 (0.49) MAPTMAPK1L3MBTL1HTTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017100668-A1 INHIBITORS OF BRUTON'S TYROSINE KINASE AND METHODS OF THEIR USE JANSSEN PHARMACEUTICA NV (BE) 2017-06-15 WO disclosed