Tiludronic Acid

Tiludronic Acid

SCHEMBL18988

O=P(O)(O)C(Sc1ccc(Cl)cc1)P(=O)(O)O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 4/20 1.00
MMP8 P22894 3/20 1.00
MMP14 P50281 2/20 1.00
MMP1 P03956 1/20 0.70
HSD17B10 Q99714 2/20 0.52
CYP2C9 P11712 1/20 0.52
CYP2C19 P33261 1/20 0.52
TSHR P16473 1/20 0.41
CA14 Q9ULX7 4/20 0.41
TRPA1 O75762 3/20 0.41
CA2 P00918 3/20 0.41
CA9 Q16790 3/20 0.41
MAPT P10636 2/20 0.41
NPSR1 Q6W5P4 2/20 0.41
CA12 O43570 2/20 0.41
CYP1A2 P05177 1/20 0.41
LMNA P02545 1/20 0.41
THRB P10828 1/20 0.41
PMP22 Q01453 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Tiludronic Acid SCHEMBL3628467 0.98 MMP2 (0.96) MMP2MMP8MMP14MMP1HSD17B10
Tiludronic Acid SCHEMBL8607914 0.96 MMP2 (0.92) MMP2MMP8MMP14MMP1HSD17B10
Tiludronic Acid SCHEMBL2067280 0.89 MMP2 (0.80) MMP2MMP8MMP14MMP1HSD17B10
SCHEMBL17954020 0.89 MMP2 (0.79) MMP2MMP8MMP14MMP1HSD17B10
Tiludronic Acid SCHEMBL7159094 0.87 MMP2 (0.77) MMP2MMP8MMP14MMP1HSD17B10
Tiludronic Acid SCHEMBL2326547 0.87 MMP2 (0.75) MMP2MMP8MMP14MMP1HSD17B10
Tiludronic Acid SCHEMBL2323298 0.87 MMP2 (0.75) MMP2MMP8MMP14MMP1HSD17B10
Tiludronic Acid SCHEMBL8607912 0.86 MMP2 (0.74) MMP2MMP8MMP14MMP1HSD17B10
Tiludronic Acid SCHEMBL41053 0.82 MMP1 (1.00) MMP2MMP8MMP14MMP1HSD17B10
Tiludronic Acid SCHEMBL8610150 0.81 MMP1 (0.96) MMP2MMP8MMP14MMP1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 16413 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3607938-B1 PHARMACEUTICAL COMPOSITION SOVIC BRKICIC LJILJANA (HR) 2026-05-27 EP claimed
US-20260137780-A1 MATERIALS AND METHODS FOR IMPROVED EXPANSION AND USES OF IMMUNE CELLS JANSSEN BIOTECH INC (US) 2026-05-21 US claimed
CN-122005812-A Combined medicine composition for engineering modification of in vivo target cells 瑞达信使(杭州)生物技术有限公司 2026-05-12 CN claimed
US-20260102414-A1 USE OF DERIVATIVES CONTAINING C-O-P BONDS IN PATIENTS WITH KIDNEY FAILURE SANIFIT THERAPEUTICS S A (ES) 2026-04-16 US claimed
US-12569507-B2 CAR T-cells for the treatment of bone metastatic cancer H. LEE MOFFITT CANCER CENTER AND RESEARCH INSTITUTE, INC. (US) 2026-03-10 US claimed
EP-4683668-A1 COMPOSITIONS AND METHODS FOR TREATING TENDON AND BONE INJURIES The United States Government as Represented by The Department of Veterans Affairs (US) 2026-01-28 EP claimed
EP-4684811-A1 NOVEL TREATMENT REGIMEN AND METHODS IN BONE HEALING Moroxite AB (SE) 2026-01-28 EP claimed
US-20250295676-A1 INOSITOL PHOSPHATE COMPOUNDS FOR USE IN TREATING, INHIBITING THE PROGRESSION, OR PREVENTING CARDIOVASCULAR CALCIFICATION VIFOR (INTERNATIONAL) LTD. (CH) 2025-09-25 US claimed
EP-3901283-B1 THERAPEUTIC TREATMENT OF BREAST CANCER BASED ON C-MAF STATUS INBIOMOTION SL (ES) 2025-08-06 EP claimed
US-12364682-B2 Use of tegaserod in preparation of anti-tumor drug QINGDAO HAIJI BIOMEDICINE CO., LTD. (CN) 2025-07-22 US claimed
EP-0600834-A1 Use of methanebisphosphonic acid derivatives for the manufacture of a medicament for fracture healing CIBA-GEIGY AG (CH) 1994-06-08 EP claimed
EP-0573604-A1 METHODS FOR THE TREATMENT OF OSTEOPOROSIS. NORWICH EATON PHARMA (US) 1993-12-15 EP claimed
EP-0550385-A1 Oral pharmaceutical compositions containing derivatives of methane-diphosphonic acid and 18-crown-6 ethers CIBA-GEIGY AG (CH) 1993-07-07 EP claimed
WO-1993011786-A1 METHODS FOR THE TREATMENT OF OSTEOPOROSIS USING BISPHOSPHONATES AND PARATHYROID HORMONE PROCTER & GAMBLE PHARMACEUTICALS, INC. (US) 1993-06-24 WO claimed
WO-1992014474-A1 METHODS FOR THE TREATMENT OF OSTEOPOROSIS NORWICH EATON PHARMACEUTICALS, INC. (US) 1992-09-03 WO claimed
US-5133972-A TOPICALLY ADMINISTRABLE PHARMACEUTICAL PREPARATIONS CIBA-GEIGY CORPORATION (US) 1992-07-28 US claimed
EP-0336851-B1 PHARMACEUTICAL COMPOSITION FOR ORAL ADMINISTRATION CONTAINING A DIPHOSPHONIC ACID DERIVATIVE ELF SANOFI (FR) 1992-03-18 EP claimed
US-4980171-A AND SODIUM LAURYL SULFATE; EXCELLENT BIOAVAILABILITY; BONE DISORSERS, ANTIARTHRETIC SOCIETE ANONYME DITE : SANOFI (FR) 1990-12-25 US claimed
EP-0276288-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING A BISPHOSPHONATE AND THEIR USE FOR NASAL ADMINISTRATION LEO PHARMACEUTICAL PRODUCTS LTD. A/S (LOVENS KEMISKE FABRIK PRODUKTIONSAKTIESELSKAB) (DK) 1988-08-03 EP claimed
WO-1988000829-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING A BISPHOSPHONATE AND THEIR USE FOR NASAL ADMINISTRATION LEO PHARMACEUTICAL PRODUCTS LTD. A/S (LØVENS KEMIS (DK) 1988-02-11 WO claimed