Tiludronic Acid

Tiludronic Acid

SCHEMBL2067280

O=P(O)(O)C(Cl)(Cl)P(=O)(O)O.O=P(O)(O)C(Sc1ccc(Cl)cc1)P(=O)(O)O

nearest known ligand 0.80

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 3/20 0.80
MMP8 P22894 2/20 0.80
MMP14 P50281 2/20 0.80
MMP1 P03956 1/20 0.58
CYP2C9 P11712 2/20 0.43
CYP2C19 P33261 2/20 0.43
HSD17B10 Q99714 1/20 0.43
TRPA1 O75762 5/20 0.41
TSHR P16473 1/20 0.39
CYP1A2 P05177 2/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CA2 P00918 2/20 0.35
CA9 Q16790 2/20 0.35
CA14 Q9ULX7 2/20 0.35
CA12 O43570 1/20 0.35
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
THRB P10828 1/20 0.35
PMP22 Q01453 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Tiludronic Acid SCHEMBL18988 0.89 MMP2 (1.00) MMP2MMP8MMP14MMP1CYP2C9
Tiludronic Acid SCHEMBL3628467 0.88 MMP2 (0.96) MMP2MMP8MMP14MMP1CYP2C9
Tiludronic Acid SCHEMBL8607914 0.86 MMP2 (0.92) MMP2MMP8MMP14MMP1CYP2C9
SCHEMBL17954020 0.79 MMP2 (0.79) MMP2MMP8MMP14MMP1CYP2C9
Tiludronic Acid SCHEMBL7159094 0.78 MMP2 (0.77) MMP2MMP8MMP14MMP1CYP2C9
Tiludronic Acid SCHEMBL2323298 0.78 MMP2 (0.75) MMP2MMP8MMP14MMP1CYP2C9
Tiludronic Acid SCHEMBL2326547 0.78 MMP2 (0.75) MMP2MMP8MMP14MMP1CYP2C9
Tiludronic Acid SCHEMBL8607912 0.77 MMP2 (0.74) MMP2MMP8MMP14MMP1CYP2C9
Tiludronic Acid SCHEMBL9850912 0.75 FDPS (0.51) MMP2MMP8MMP14MMP1CYP2C9
Tiludronic Acid SCHEMBL41053 0.74 MMP1 (1.00) MMP2MMP8MMP14MMP1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240174665-A1 CDK2 INHIBITORS AND USES THEREOF KYMERA THERAPEUTICS, INC. 2024-05-30 US disclosed
US-20240173419-A1 CDK2 DEGRADERS AND USES THEREOF KYMERA THERAPEUTICS, INC. 2024-05-30 US disclosed
US-20230110180-A1 CDK2 DEGRADERS AND USES THEREOF KYMERA THERAPEUTICS, INC. 2023-04-13 US disclosed
US-10266535-B2 Inhibitor of FLT3 kinase and use thereof HEFEI INSTITUTES OF PHYSICAL SCIENCE, CHINESE ACADEMY OF SCIENCES (CN) 2019-04-23 US disclosed
US-20180030054-A1 NOVEL INHIBITOR OF FLT3 KINASE AND USE THEREOF HEFEI INSTITUTES OF PHYSICAL SCIENCE, CHINESE ACADEMY OF SCIENCES (CN) 2018-02-01 US disclosed
EP-2438064-A1 1H-IMIDAZO[4,5-c]QUINOLINONE DERIVATIVES Novartis AG (CH) 2012-04-11 EP disclosed
WO-2010139731-A1 1H-IMIDAZO[4,5-c]QUINOLINONE DERIVATIVES NOVARTIS AG (CH) 2010-12-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240174665-A1 CDK2 INHIBITORS AND USES THEREOF CDK2, CDK20, CDK1 MMP2 2855/4885MMP8 3521/4885MMP14 2408/4885
US-20180030054-A1 NOVEL INHIBITOR OF FLT3 KINASE AND USE THEREOF FLT3, FLT1, FGFR1 MMP2 3227/4885MMP8 4114/4885MMP14 2673/4885
US-20230110180-A1 CDK2 DEGRADERS AND USES THEREOF CDK2, CDK20, CDK1 MMP2 1416/4885MMP8 2855/4885MMP14 980/4885
US-20240173419-A1 CDK2 DEGRADERS AND USES THEREOF CDK2, CDK20, CDK1 MMP2 1416/4885MMP8 2855/4885MMP14 980/4885
US-10266535-B2 Inhibitor of FLT3 kinase and use thereof FLT3, FLT1, FGFR1 MMP2 3121/4885MMP8 4070/4885MMP14 2591/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.