SCHEMBL19003300

SCHEMBL19003300

O=C(/C=C/c1ccc(-c2ccccc2)s1)Nc1ccc(-c2nnco2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 1/20 0.45
HSD17B2 P37059 1/20 0.45
NOTUM Q6P988 1/20 0.44
MAPT P10636 4/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
MAPK1 P28482 1/20 0.39
TSHR P16473 1/20 0.39
TLR8 Q9NR97 1/20 0.38
HTT P42858 2/20 0.38
NPC1 O15118 2/20 0.38
MEN1 O00255 1/20 0.38
LMNA P02545 1/20 0.38
KMT2A Q03164 1/20 0.38
MMP1 P03956 5/20 0.38
MMP2 P08253 5/20 0.38
MMP9 P14780 5/20 0.38
EGFR P00533 4/20 0.38
RAB9A P51151 2/20 0.38
MAOA P21397 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19003249 0.84 EGFR (0.42) NOTUMMAPTTSHRHTTNPC1
SCHEMBL19003343 0.79 MAPT (0.46) NOTUMMAPTKDM4EALDH1A1MAPK1
SCHEMBL18985528 0.79 NQO2 (0.56) HSD17B1HSD17B2MAPTKDM4EALDH1A1
SCHEMBL19003466 0.79 NQO2 (0.56) HSD17B1HSD17B2MAPTKDM4EALDH1A1
SCHEMBL19003299 0.77 MAPT (0.52) HSD17B1HSD17B2MAPTKDM4EALDH1A1
SCHEMBL19003302 0.77 HSD17B1 (0.48) HSD17B1HSD17B2MAPTKDM4EALDH1A1
SCHEMBL19003306 0.76 TRPV1 (0.61) HSD17B1HSD17B2NOTUMMAPTKDM4E
SCHEMBL19003303 0.76 MAOB (0.52) HSD17B1HSD17B2MAPTALDH1A1HTT
SCHEMBL18985199 0.75 NAMPT (0.48) HSD17B1HSD17B2MAPTKDM4EALDH1A1
SCHEMBL19003304 0.74 ABL1 (0.58) MAPTKDM4EALDH1A1NPC1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017102014-A1 PROPENAMIDE THIOPHENE DERIVATIVES AS FLAVIVIRUS INHIBITORS AND THEIR USE UNIVERSITE D'AIX-MARSEILLE (FR) 2017-06-22 WO disclosed