SCHEMBL19003306

SCHEMBL19003306

O=C(CCc1ccc(-c2ccccc2)s1)Nc1ccc(-c2nnco2)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 5/20 0.61
HSD17B1 P14061 1/20 0.46
HSD17B2 P37059 1/20 0.46
NOTUM Q6P988 1/20 0.45
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
TNKS O95271 1/20 0.43
TNKS2 Q9H2K2 1/20 0.43
HPGD P15428 4/20 0.43
ESR1 P03372 1/20 0.43
POLB P06746 1/20 0.43
MAPT P10636 1/20 0.43
KDM4E B2RXH2 2/20 0.42
HSD17B10 Q99714 2/20 0.42
TSHR P16473 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
ALDH1A1 P00352 1/20 0.42
PKM P14618 1/20 0.42
USP2 O75604 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19003300 0.76 HSD17B1 (0.45) TRPV1HSD17B1HSD17B2NOTUMNPC1
SCHEMBL9002868 0.74 TRPV1 (0.58) TRPV1HSD17B1HSD17B2NPC1RAB9A
SCHEMBL14340845 0.72 HCAR2 (0.67) TRPV1NPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL19003343 0.72 MAPT (0.46) NOTUMHPGDMAPTKDM4EHSD17B10
SCHEMBL29236054 0.72 NOTUM (0.56) TRPV1NOTUMHPGDESR1POLB
SCHEMBL3182274 0.72 TRPV1 (0.55) TRPV1HSD17B1HSD17B2HPGDMAPT
SCHEMBL4619799 0.69 RPS6KB2 (0.60) TRPV1RAB9APOLBMAPTHSD17B10
SCHEMBL29235975 0.69 TSHR (0.58) NOTUMHPGDESR1POLBMAPT
SCHEMBL17205531 0.67 TRPV1 (1.00) TRPV1
SCHEMBL5571187 0.67 NOTUM (0.91) NOTUMMAPTKDM4ETSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017102014-A1 PROPENAMIDE THIOPHENE DERIVATIVES AS FLAVIVIRUS INHIBITORS AND THEIR USE UNIVERSITE D'AIX-MARSEILLE (FR) 2017-06-22 WO disclosed