SCHEMBL19003364

SCHEMBL19003364

O=C(/C=C/c1ccc(Br)s1)Nc1cnc2ccccc2c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 7/20 0.49
EGFR P00533 1/20 0.48
KDM4E B2RXH2 5/20 0.48
NPC1 O15118 6/20 0.47
RAB9A P51151 6/20 0.47
SMN1; SMN2 Q16637 4/20 0.47
HSD17B10 Q99714 3/20 0.47
TP53 P04637 1/20 0.47
POLB P06746 2/20 0.46
MAPT P10636 1/20 0.46
ALDH1A1 P00352 1/20 0.46
NAMPT P43490 1/20 0.46
USP30 Q70CQ3 1/20 0.46
HDAC3 O15379 1/20 0.46
HDAC4 P56524 1/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC7 Q8WUI4 1/20 0.46
HDAC2 Q92769 1/20 0.46
HDAC10 Q969S8 1/20 0.46
HDAC11 Q96DB2 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16101601 0.79 KDR (0.60) KDREGFRKDM4ENPC1RAB9A
SCHEMBL13991500 0.79 KDR (0.60) KDREGFRKDM4ENPC1RAB9A
SCHEMBL879570 0.76 KDM4E (0.62) KDRKDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL13991503 0.75 RAB9A (0.65) KDREGFRKDM4ENPC1RAB9A
SCHEMBL18985272 0.74 MAOB (0.63) EGFRNPC1RAB9ASMN1; SMN2TP53
SCHEMBL19003356 0.74 TRPV1 (0.49) EGFRNPC1RAB9ASMN1; SMN2MAPT
SCHEMBL846549 0.74 DHODH (0.53) KDRKDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL846550 0.74 DHODH (0.53) KDRKDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL29965933 0.73 KDR (0.62) KDRKDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL4018954 0.73 KDR (0.62) KDRKDM4ENPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017102014-A1 PROPENAMIDE THIOPHENE DERIVATIVES AS FLAVIVIRUS INHIBITORS AND THEIR USE UNIVERSITE D'AIX-MARSEILLE (FR) 2017-06-22 WO disclosed