SCHEMBL19003356

SCHEMBL19003356

O=C(/C=C/c1ccc(Br)s1)Nc1cncc2ccccc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 2/20 0.49
CHEK1 O14757 1/20 0.49
PIM1 P11309 1/20 0.49
CDK8 P49336 1/20 0.49
GSK3B P49841 1/20 0.49
CDK7 P50613 1/20 0.49
CDK9 P50750 1/20 0.49
LIMK1 P53667 1/20 0.49
ROCK1 Q13464 1/20 0.49
CLK4 Q9HAZ1 1/20 0.49
EGFR P00533 2/20 0.41
HDAC1 Q13547 4/20 0.41
HDAC2 Q92769 3/20 0.41
RAB9A P51151 5/20 0.40
SMN1; SMN2 Q16637 5/20 0.40
NPC1 O15118 4/20 0.40
LMNA P02545 2/20 0.40
MEN1 O00255 2/20 0.40
MAPT P10636 2/20 0.40
KMT2A Q03164 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19003261 0.75 MMP1 (0.59) EGFRHDAC1HDAC2RAB9ASMN1; SMN2
SCHEMBL19003357 0.74 EGFR (0.42) EGFRRAB9ASMN1; SMN2NPC1LMNA
SCHEMBL19003364 0.74 KDR (0.49) EGFRHDAC1HDAC2RAB9ASMN1; SMN2
SCHEMBL19003354 0.72 MMP1 (0.62) TRPV1EGFRHDAC1HDAC2RAB9A
SCHEMBL19003351 0.71 LMNA (0.50) EGFRRAB9ASMN1; SMN2NPC1LMNA
SCHEMBL19003363 0.70 RAB9A (0.52) EGFRRAB9ASMN1; SMN2NPC1LMNA
SCHEMBL27034898 0.69 KDM4E (0.62) TRPV1RAB9ASMN1; SMN2NPC1MEN1
SCHEMBL14665804 0.68 ADRA2A (0.50) MEN1MAPTKMT2AHDAC6MALT1
SCHEMBL18985272 0.68 MAOB (0.63) TRPV1EGFRRAB9ASMN1; SMN2NPC1
SCHEMBL19003255 0.68 EGFR (0.47) EGFRRAB9ASMN1; SMN2NPC1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017102014-A1 PROPENAMIDE THIOPHENE DERIVATIVES AS FLAVIVIRUS INHIBITORS AND THEIR USE UNIVERSITE D'AIX-MARSEILLE (FR) 2017-06-22 WO disclosed