SCHEMBL19004853

SCHEMBL19004853

COc1c(N)ncnc1NC1CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 12/20 0.43
CYP1A2 P05177 3/20 0.41
CYP3A4 P08684 3/20 0.41
CYP2D6 P10635 3/20 0.41
USP2 O75604 2/20 0.41
LMNA P02545 2/20 0.41
TSHR P16473 2/20 0.41
CYP2C19 P33261 2/20 0.41
CLK4 Q9HAZ1 2/20 0.41
ALDH1A1 P00352 1/20 0.41
ALOX15 P16050 1/20 0.41
MAPK1 P28482 1/20 0.41
HPGDS O60760 2/20 0.40
EGFR P00533 1/20 0.39
PDE5A O76074 1/20 0.37
TP53 P04637 1/20 0.37
POLB P06746 1/20 0.37
PKM P14618 1/20 0.37
NFKB1 P19838 1/20 0.37
ADORA1 P30542 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19004849 0.94 HPGDS (0.44) IRAK4CYP1A2CYP3A4CYP2D6LMNA
SCHEMBL19005056 0.83 HPGDS (0.40) IRAK4LMNAHPGDSEGFRPKM
SCHEMBL19004855 0.76 BTK (0.40) EGFR
SCHEMBL22897343 0.75 EGFR (0.44) CYP1A2CYP3A4CYP2D6LMNAHPGDS
SCHEMBL17369356 0.74 GSK3B (0.46) TSHRALDH1A1
SCHEMBL23555498 0.74 IRAK4 (0.44) IRAK4CYP1A2CYP3A4CYP2D6LMNA
SCHEMBL28890932 0.74 HPGDS (0.42) IRAK4CYP3A4LMNAHPGDSEGFR
SCHEMBL24344303 0.73 IRAK4 (0.43) IRAK4CYP1A2CYP3A4CYP2D6USP2
SCHEMBL29534716 0.73 IRAK4 (0.43) IRAK4CYP1A2CYP3A4CYP2D6USP2
SCHEMBL24344307 0.71 CYP3A4 (0.45) IRAK4CYP1A2CYP3A4CYP2D6USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017102091-A1 HETEROARYLBENZIMIDAZOLE COMPOUNDS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2017-06-22 WO disclosed