SCHEMBL19004855

SCHEMBL19004855

COc1c(N)ncnc1NCC1CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BTK Q06187 8/20 0.40
TRPM8 Q7Z2W7 1/20 0.39
FFAR2 O15552 1/20 0.38
PIK3CD O00329 1/20 0.38
ADORA2A P29274 1/20 0.38
PDE10A Q9Y233 1/20 0.38
GRM1 Q13255 1/20 0.38
HRH4 Q9H3N8 1/20 0.38
STK4 Q13043 1/20 0.37
STK3 Q13188 1/20 0.37
EGFR P00533 1/20 0.36
TEC P42680 1/20 0.36
BMX P51813 1/20 0.36
CD69 Q07108 1/20 0.36
ITK Q08881 1/20 0.36
KCNH2 Q12809 1/20 0.36
ERBB4 Q15303 1/20 0.36
GP6 Q9HCN6 1/20 0.36
NUDT5 Q9UKK9 1/20 0.36
KHK P50053 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19004853 0.76 IRAK4 (0.43) EGFR
SCHEMBL26496338 0.75 USP7 (0.41) BTKFFAR2ADORA2APDE10AHRH4
SCHEMBL19004849 0.74 HPGDS (0.44) ADORA2AEGFRJAK2JAK1
SCHEMBL25075340 0.71 BTK (0.36) BTKFFAR2PIK3CDADORA2APDE10A
SCHEMBL26493919 0.71 BTK (0.36) BTKFFAR2ADORA2APDE10AHRH4
SCHEMBL20732651 0.71 TRPM8 (0.51) TRPM8PDE10AKHK
SCHEMBL17369356 0.71 GSK3B (0.46)
SCHEMBL12590817 0.70 RAB9A (0.48) FFAR2PDE10AHRH4STK4STK3
SCHEMBL14241098 0.68 AURKA (0.49) FFAR2STK4STK3KHKJAK2
SCHEMBL26493925 0.67 BTK (0.41) BTKEGFRTECBMXCD69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017102091-A1 HETEROARYLBENZIMIDAZOLE COMPOUNDS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2017-06-22 WO disclosed