SCHEMBL19005732

SCHEMBL19005732

c1cn2c(n1)CCC1CNCCC12

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 9/20 0.33
CHRNB4 P30926 9/20 0.33
CHRNA3 P32297 9/20 0.33
CHRNA4 P43681 9/20 0.33
ADRA1A P35348 1/20 0.31
HTR2A P28223 1/20 0.30
HTR2C P28335 1/20 0.30
HTR2B P41595 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19005804 0.75 CHRNB2 (0.31) CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL19005688 0.75 CHRNB2 (0.31) CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL19005659 0.75 CHRNB2 (0.31) CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL19005657 0.72 CHRNB2 (0.34) CHRNB2CHRNB4CHRNA3CHRNA4HTR2A
SCHEMBL19005651 0.71 SIGMAR1 (0.36) ADRA1A
SCHEMBL19005658 0.71 ADRA1A (0.33) ADRA1A
SCHEMBL19005642 0.70 SLC18A3 (0.35) CHRNB2CHRNB4CHRNA3CHRNA4HTR2A
SCHEMBL19005648 0.69 CYP19A1 (0.40) CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL19005645 0.66 MEN1 (0.41) CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL13755325 0.65

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017101796-A1 PHTHALAZINONE DERIVATIVE, AND PREPARATION METHOD AND USE THEREOF 四川科伦博泰生物医药股份有限公司 2017-06-22 WO disclosed