SCHEMBL19005733

SCHEMBL19005733

CN1CCCC2C1CCc1cccn12

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CHRNB4 P30926 3/20 0.40
CHRNA3 P32297 3/20 0.40
CHRNB2 P17787 2/20 0.40
CHRNA4 P43681 2/20 0.40
CHRNA7 P36544 1/20 0.40
DRD2 P14416 2/20 0.37
L3MBTL3 Q96JM7 1/20 0.36
CHRM2 P08172 4/20 0.36
CHRM4 P08173 4/20 0.36
CHRM5 P08912 4/20 0.36
CHRM1 P11229 4/20 0.36
CHRM3 P20309 4/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19005649 0.73 CYP19A1 (0.42) CHRNB4CHRNA3
SCHEMBL2274269 0.72 CHRM2 (0.45) CHRNB4CHRNA3CHRNB2CHRNA4CHRNA7
SCHEMBL20384062 0.72 CHRM2 (0.45) CHRNB4CHRNA3CHRNB2CHRNA4CHRNA7
SCHEMBL19005734 0.70 CHRNB4 (0.35) CHRNB4CHRNA3CHRNB2CHRNA4
SCHEMBL19005643 0.70 CHRNB4 (0.39) CHRNB4CHRNA3CHRNB2CHRNA4CHRNA7
SCHEMBL10092844 0.70
SCHEMBL19005661 0.68 DRD2 (0.37) DRD2L3MBTL3
SCHEMBL20939371 0.68 CHRM2 (0.47) CHRNB4CHRNA3CHRNB2CHRNA4CHRNA7
SCHEMBL17888212 0.68 ALDH1A1 (0.45) CHRNB4CHRNA3CHRNB2CHRNA4CHRNA7
SCHEMBL19992145 0.68 CHRM2 (0.47) CHRNB4CHRNA3CHRNB2CHRNA4CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017101796-A1 PHTHALAZINONE DERIVATIVE, AND PREPARATION METHOD AND USE THEREOF 四川科伦博泰生物医药股份有限公司 2017-06-22 WO disclosed