SCHEMBL19005997

SCHEMBL19005997

CCCOc1cc2c(cc1C(O)CCc1ccc(OC)c(N)c1)OCS2(=O)=O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.34
KCNH2 Q12809 2/20 0.34
TMEM97 Q5BJF2 1/20 0.34
ADRB2 P07550 2/20 0.34
ADRB1 P08588 2/20 0.34
ADRB3 P13945 2/20 0.34
GAA P10253 2/20 0.33
ADRA1D P25100 1/20 0.33
ADRA1A P35348 1/20 0.33
ADRA1B P35368 1/20 0.33
STAT3 P40763 1/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
KDM4E B2RXH2 1/20 0.32
USP2 O75604 1/20 0.32
ALDH1A1 P00352 1/20 0.32
TP53 P04637 1/20 0.32
POLB P06746 1/20 0.32
MAPT P10636 1/20 0.32
CASP1 P29466 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19006007 0.90 CYP3A4 (0.39) SIGMAR1KCNH2TMEM97ADRB2GAA
SCHEMBL18987263 0.90 KCNH2 (0.34) SIGMAR1KCNH2TMEM97STAT3KDM4E
SCHEMBL18987234 0.84 PPARG (0.32) PPARGPPARA
SCHEMBL19005915 0.84 PDE4A (0.33) ADRB2ADRB1ADRB3ADRA1DADRA1A
SCHEMBL19005966 0.82 CYP3A4 (0.38) SIGMAR1KCNH2TMEM97GAAMEN1
SCHEMBL19005967 0.82 GAA (0.36) GAAMEN1KMT2AKDM4EUSP2
SCHEMBL19005989 0.81 HDAC1 (0.37) SIGMAR1KCNH2GAAMEN1KMT2A
SCHEMBL19005987 0.78 HDAC1 (0.38) GAAMEN1KMT2AKDM4EALDH1A1
SCHEMBL19005918 0.73 HTR1A (0.38) SIGMAR1KCNH2TMEM97GAAMEN1
SCHEMBL19005956 0.73 HTR1A (0.36) SIGMAR1KCNH2GAAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017103637-A1 DIPHENYLPROPANE COMPOUNDS AND THEIR CYTOTOXIC ACTIVITY BLIRT S.A. (PL) 2017-06-22 WO disclosed