SCHEMBL19005987

SCHEMBL19005987

CCCOc1cc2c(cc1C(N)CCc1ccc(OC)c(NC(=O)CCC)c1)OCS2(=O)=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 3/20 0.38
HDAC2 Q92769 3/20 0.38
MEN1 O00255 2/20 0.36
CYP1A2 P05177 2/20 0.36
KMT2A Q03164 2/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
TSHR P16473 1/20 0.36
CYP2C19 P33261 1/20 0.36
LTB4R Q15722 1/20 0.35
POLB P06746 2/20 0.35
GAA P10253 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
ALDH1A1 P00352 3/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
KDM4E B2RXH2 2/20 0.34
HPGD P15428 2/20 0.34
HSD17B10 Q99714 2/20 0.34
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19005966 0.86 CYP3A4 (0.38) MEN1CYP1A2KMT2ACYP3A4TSHR
SCHEMBL19005915 0.84 PDE4A (0.33) HDAC1HDAC2TSHRSMN1; SMN2MAPT
SCHEMBL19005992 0.79 HDAC1 (0.39) HDAC1HDAC2MEN1CYP1A2KMT2A
SCHEMBL19006008 0.79 HDAC1 (0.36) HDAC1HDAC2MEN1CYP1A2KMT2A
SCHEMBL19005997 0.78 SIGMAR1 (0.34) HDAC1HDAC2MEN1CYP1A2KMT2A
SCHEMBL19005991 0.78 MTNR1A (0.34) HDAC1HDAC2KMT2ATSHRPOLB
SCHEMBL19006007 0.77 CYP3A4 (0.39) MEN1CYP1A2KMT2ACYP3A4TSHR
SCHEMBL18987263 0.76 KCNH2 (0.34) ALDH1A1KDM4E
SCHEMBL19005989 0.72 HDAC1 (0.37) HDAC1HDAC2MEN1CYP1A2KMT2A
SCHEMBL19006005 0.70 HTR1A (0.34) HDAC1HDAC2TSHRPOLBSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017103637-A1 DIPHENYLPROPANE COMPOUNDS AND THEIR CYTOTOXIC ACTIVITY BLIRT S.A. (PL) 2017-06-22 WO disclosed