SCHEMBL19005915

SCHEMBL19005915

CCCOc1cc2c(cc1C(O)CCc1ccc(OC)c(NC(=O)[C@@H](N)CC)c1)OCS2(=O)=O

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 2/20 0.33
PDE4B Q07343 2/20 0.33
PDE4C Q08493 2/20 0.33
PDE4D Q08499 2/20 0.33
HDAC1 Q13547 1/20 0.32
HDAC2 Q92769 1/20 0.32
ADRB2 P07550 2/20 0.32
ADRB1 P08588 2/20 0.32
ADRB3 P13945 2/20 0.32
LNPEP Q9UIQ6 3/20 0.32
PPARA Q07869 2/20 0.32
MAPT P10636 1/20 0.32
TSHR P16473 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
REN P00797 1/20 0.31
LMNA P02545 1/20 0.31
MAPK1 P28482 1/20 0.31
AAK1 Q2M2I8 1/20 0.31
ADRA1D P25100 1/20 0.31
ADRA1A P35348 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19005991 0.86 MTNR1A (0.34) PDE4APDE4BPDE4CPDE4DHDAC1
SCHEMBL19006008 0.86 HDAC1 (0.36) HDAC1HDAC2PPARAMAPTTSHR
SCHEMBL19005997 0.84 SIGMAR1 (0.34) PDE4APDE4BPDE4CPDE4DHDAC1
SCHEMBL19005987 0.84 HDAC1 (0.38) HDAC1HDAC2MAPTTSHRSMN1; SMN2
SCHEMBL19006007 0.83 CYP3A4 (0.39) ADRB2TSHRLMNA
SCHEMBL18987263 0.82 KCNH2 (0.34) PDE4D
SCHEMBL19006005 0.79 HTR1A (0.34) PDE4APDE4BPDE4CPDE4DHDAC1
SCHEMBL19005966 0.78 CYP3A4 (0.38) MAPTTSHRLMNA
SCHEMBL18987234 0.75 PPARG (0.32) PPARATSHRLMNAPPARG
SCHEMBL19005992 0.74 HDAC1 (0.39) PDE4APDE4BPDE4CPDE4DHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017103637-A1 DIPHENYLPROPANE COMPOUNDS AND THEIR CYTOTOXIC ACTIVITY BLIRT S.A. (PL) 2017-06-22 WO disclosed