SCHEMBL19006770

SCHEMBL19006770

Cc1cnc2n1-c1ccc(Cl)cc1C(c1ccccn1)=NC2

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 5/20 0.55
GABRA5 P31644 5/20 0.55
GABRA3 P34903 5/20 0.55
GABRA2 P47869 5/20 0.55
GABRB2 P47870 4/20 0.55
CYP1A2 P05177 1/20 0.53
OPRK1 P41145 6/20 0.51
HPGD P15428 4/20 0.51
LMNA P02545 2/20 0.51
BRD4 O60885 2/20 0.51
CNR1 P21554 1/20 0.51
PDE4D Q08499 3/20 0.50
GABRG2 P18507 2/20 0.50
GABRB3 P28472 2/20 0.50
HTR2A P28223 1/20 0.50
ADRA1A P35348 1/20 0.50
CYP3A4 P08684 2/20 0.47
SLC22A1 O15245 1/20 0.47
ABCB11 O95342 1/20 0.47
DRD3 P35462 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11827431 0.90 OPRK1 (0.51) GABRA1GABRA5GABRA3GABRA2GABRB2
SCHEMBL22591865 0.88 GABRA3 (0.51) GABRA1GABRA5GABRA3GABRA2GABRB2
SCHEMBL11828965 0.87 GABRA3 (0.73) GABRA1GABRA5GABRA3GABRA2GABRB2
SCHEMBL29783033 0.87 GABRA3 (0.73) GABRA1GABRA5GABRA3GABRA2GABRB2
SCHEMBL11809246 0.85 OPRK1 (0.69) GABRA1GABRA5GABRA3GABRA2GABRB2
SCHEMBL22591822 0.85 GABRA3 (0.53) GABRA1GABRA5GABRA3GABRA2GABRB2
SCHEMBL11620342 0.84 GABRA1 (0.77) GABRA1GABRA5GABRA3GABRA2GABRB2
SCHEMBL11825295 0.84 GABRA1 (0.70) GABRA1GABRA5GABRA3GABRA2GABRB2
SCHEMBL24383773 0.84 GABRA1 (0.53) GABRA1GABRA5GABRA3GABRA2GABRB2
SCHEMBL24383816 0.84 GABRA1 (0.50) GABRA1GABRA5GABRA3GABRA2GABRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017101808-A1 SHORT-ACTING BENZODIAZEPINE DERIVATIVE, PREPARATION METHOD THEREFOR, AND USE THEREOF 四川科伦博泰生物医药股份有限公司 2017-06-22 WO disclosed