SCHEMBL19019155

SCHEMBL19019155

O=c1[nH]c2ccc(S(=O)(=O)Nc3ccc(Br)cc3)cc2[nH]c1=O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.84
IDO1 P14902 1/20 0.63
PKM P14618 4/20 0.62
MEN1 O00255 1/20 0.62
KMT2A Q03164 1/20 0.62
TAS2R14 Q9NYV8 1/20 0.59
ALDH1A1 P00352 1/20 0.58
MAPT P10636 3/20 0.56
MAPK1 P28482 1/20 0.55
TP53 P04637 1/20 0.54
NPSR1 Q6W5P4 1/20 0.52
PGR P06401 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19018960 0.85 POLB (0.64) POLBPKMMEN1KMT2ATAS2R14
SCHEMBL22425031 0.82 POLB (0.84) POLBIDO1PKMMEN1KMT2A
SCHEMBL19019156 0.82 MAPT (0.67) POLBPKMMEN1KMT2ATAS2R14
SCHEMBL24876169 0.77 MEN1 (0.72) POLBPKMMEN1KMT2AMAPT
SCHEMBL9535518 0.77 NPSR1 (0.65) POLBIDO1PKMMEN1KMT2A
SCHEMBL26597984 0.77 KMT2A (0.74) POLBPKMMEN1KMT2AALDH1A1
SCHEMBL1279534 0.74 TAS2R14 (1.00) POLBPKMMEN1KMT2ATAS2R14
SCHEMBL24430215 0.74 POLB (0.71) POLBIDO1PKMMEN1KMT2A
SCHEMBL31680036 0.74 THRB (0.58) POLBPKMMEN1KMT2AALDH1A1
SCHEMBL18173883 0.73 MAPT (0.79) POLBPKMMEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10208000-B2 Eis inhibitors UNIVERSITY OF KENTUCKY RESEARCH FOUNDATION (US) 2019-02-19 US disclosed
US-20170174639-A1 EIS INHIBITORS UNIVERSITY OF KENTUCKY RESEARCH FOUNDATION 2017-06-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170174639-A1 EIS INHIBITORS ABCC1, ATP5ME, ABCG2 POLB 1092/4885IDO1 2014/4885PKM 624/4885
US-10208000-B2 Eis inhibitors ABCC1, ATP5ME, ABCG2 POLB 1092/4885IDO1 2014/4885PKM 624/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.