SCHEMBL1905233

SCHEMBL1905233

CN1CCC[C@@H]1C(=O)N[C@@H](Cc1cccc2ccccc12)C(=O)NCc1cnc(N)s1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NTMT1 Q9BV86 2/20 0.44
TACR1 P25103 3/20 0.43
FNTA P49354 1/20 0.41
PGGT1B P53609 1/20 0.41
P2RX7 Q99572 1/20 0.40
MMP2 P08253 1/20 0.38
MMP9 P14780 1/20 0.38
MMP8 P22894 1/20 0.38
LCK P06239 1/20 0.38
CTSS P25774 1/20 0.38
CTSK P43235 1/20 0.38
MC4R P32245 2/20 0.37
MC1R Q01726 2/20 0.37
MC3R P41968 1/20 0.37
DPP4 P27487 1/20 0.37
PLG P00747 1/20 0.37
PRSS1 P07477 1/20 0.37
PRSS2 P07478 1/20 0.37
PRSS3 P35030 1/20 0.37
OPRD1 P41143 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1906955 1.00 NTMT1 (0.44) NTMT1TACR1FNTAPGGT1BP2RX7
SCHEMBL1904935 0.90 TACR1 (0.41) NTMT1TACR1DPP4
SCHEMBL1902611 0.90 TACR1 (0.41) NTMT1TACR1DPP4
SCHEMBL1903923 0.89 TACR1 (0.41) TACR1DPP4
SCHEMBL1908359 0.89 TACR1 (0.41) TACR1DPP4
SCHEMBL1433336 0.86 TACR1 (0.46) NTMT1TACR1FNTAPGGT1BP2RX7
SCHEMBL1906919 0.83 CTSB (0.40) CTSSCTSK
SCHEMBL13623819 0.83 F2 (0.52) NTMT1TACR1P2RX7
SCHEMBL1432873 0.83 F2 (0.52) NTMT1TACR1P2RX7
SCHEMBL1901984 0.83 MEN1 (0.39) TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011051673-A1 AMINOTHIAZOLE DERIVATIVES USEFUL AS KLK1 INHIBITORS VANTIA LIMITED (GB) 2011-05-05 WO disclosed