SCHEMBL1905802

SCHEMBL1905802

CN1CCC[C@@H]1C(=O)N[C@@H](Cc1cccc(Cl)c1)C(=O)NCc1cnc(N)s1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CTSL P07711 16/20 0.47
CTSS P25774 16/20 0.47
CTSV O60911 15/20 0.47
CTSK P43235 12/20 0.47
CTSB P07858 9/20 0.43
F2 P00734 2/20 0.42
ADAM17 P78536 1/20 0.40
ITGB1 P05556 1/20 0.40
ITGA4 P13612 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1906106 1.00 CTSL (0.47) CTSLCTSSCTSVCTSKCTSB
SCHEMBL1906919 0.91 CTSB (0.40) CTSLCTSSCTSVCTSKCTSB
SCHEMBL1906321 0.91 KMT2A (0.41) CTSLCTSSCTSVCTSK
SCHEMBL1908228 0.91 KMT2A (0.41) CTSLCTSSCTSVCTSK
SCHEMBL1904713 0.90 LCK (0.39) ITGB1ITGA4
SCHEMBL1905914 0.90 TACR1 (0.43) CTSLITGB1ITGA4
SCHEMBL1905803 0.90 TACR1 (0.43) CTSLITGB1ITGA4
SCHEMBL1902249 0.89 MEN1 (0.39)
SCHEMBL1905042 0.89 MEN1 (0.39)
SCHEMBL1904624 0.89 MEN1 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011051673-A1 AMINOTHIAZOLE DERIVATIVES USEFUL AS KLK1 INHIBITORS VANTIA LIMITED (GB) 2011-05-05 WO claimed
WO-2011051673-A1 AMINOTHIAZOLE DERIVATIVES USEFUL AS KLK1 INHIBITORS VANTIA LIMITED (GB) 2011-05-05 WO disclosed