SCHEMBL19066913

SCHEMBL19066913

Cc1cc(N)sc1C(=O)OC(C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CISD2 Q8N5K1 1/20 0.42
GRM6 O15303 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.39
NPC1 O15118 1/20 0.39
HTT P42858 1/20 0.39
RAB9A P51151 1/20 0.39
MAPK14 Q16539 1/20 0.37
ALOX15 P16050 2/20 0.36
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
LHCGR P22888 1/20 0.34
LCK P06239 2/20 0.34
ALDH1A1 P00352 5/20 0.33
KDM4E B2RXH2 2/20 0.33
GAA P10253 2/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL381164 0.80 MAPK14 (0.52) CISD2NPC1RAB9AMAPK14ALOX15
SCHEMBL20263505 0.79 NPC1 (0.39) CISD2GRM6SMN1; SMN2NPC1HTT
SCHEMBL2434324 0.79 NPC1 (0.40) CISD2GRM6SMN1; SMN2NPC1HTT
Hydrochloric Acid SCHEMBL5445499 0.79 MAPK14 (0.51) CISD2NPC1RAB9AMAPK14ALOX15
SCHEMBL244336 0.77 ALOX15 (0.58) SMN1; SMN2NPC1HTTRAB9AALOX15
Hydrochloric Acid SCHEMBL244320 0.76 ALOX15 (0.56) SMN1; SMN2NPC1HTTRAB9AALOX15
SCHEMBL7264963 0.75 GRM6 (0.51) GRM6SMN1; SMN2NPC1RAB9ALHCGR
SCHEMBL14029306 0.74 KDM4E (0.45) CISD2SMN1; SMN2NPC1HTTRAB9A
SCHEMBL243572 0.74 KDM4E (0.42) SMN1; SMN2NPC1RAB9AMAPK14ALOX15
SCHEMBL14507422 0.74 IKBKB (0.45) ALOX15CYP2C9ALDH1A1GAAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20190010144-A1 SMALL MOLECULE INHIBITOR OF 3-PHOSPHOGLYCERATE DEHYDROGENASE AND USES THEREOF CORNELL UNIVERSITY 2019-01-10 US disclosed
WO-2017117532-A1 SMALL MOLECULE INHIBITOR OF 3-PHOSPHOGLYCERATE DEHYDROGENASE AND USES THEREOF CANTLEY LEWIS C (US) 2017-07-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190010144-A1 SMALL MOLECULE INHIBITOR OF 3-PHOSPHOGLYCERATE DEHYDROGENASE AND USES THEREOF PHGDH, G6PD, PGD CISD2 269/4885GRM6 1805/4885SMN1; SMN2 4245/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.