SCHEMBL1907892

SCHEMBL1907892

Nc1ncc(CNC(=O)C(N)Cc2cccc3ccccc23)s1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 2/20 0.46
ROCK2 O75116 1/20 0.46
PIM1 P11309 1/20 0.46
PRKACA P17612 1/20 0.46
FGFR3 P22607 1/20 0.46
GSK3A P49840 1/20 0.46
RPS6KA3 P51812 1/20 0.46
LIMK1 P53667 1/20 0.46
PRKCD Q05655 1/20 0.46
ROCK1 Q13464 1/20 0.46
DYRK1A Q13627 1/20 0.46
CDC42BPA Q5VT25 1/20 0.46
SIRT2 Q8IXJ6 2/20 0.41
COPS5 Q92905 1/20 0.41
NLN Q9BYT8 2/20 0.41
SLC1A3 P43003 1/20 0.40
SLC1A2 P43004 1/20 0.40
SLC1A1 P43005 1/20 0.40
ATG4B Q9Y4P1 1/20 0.40
LMNA P02545 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1907890 1.00 AKT1 (0.46) AKT1ROCK2PIM1PRKACAFGFR3
Trifluoroacetic Acid SCHEMBL1906333 0.93 DRD2 (0.44) AKT1ROCK2PIM1PRKACAFGFR3
SCHEMBL1905660 0.82 MME (0.51) SIRT2
SCHEMBL1905678 0.81 MME (0.43) SIRT2
SCHEMBL3146169 0.81 MASP2 (0.48) AKT1ROCK2PIM1PRKACAFGFR3
Hydrochloric Acid SCHEMBL1902944 0.80 MASP2 (0.48) AKT1ROCK2PIM1PRKACAFGFR3
SCHEMBL1908220 0.80 CTSS (0.64)
SCHEMBL6901592 0.80 CTSS (0.39) SIRT2
SCHEMBL7860770 0.80 EGFR (0.53) AKT1ROCK2PIM1PRKACAFGFR3
SCHEMBL7860766 0.80 EGFR (0.53) AKT1ROCK2PIM1PRKACAFGFR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011051673-A1 AMINOTHIAZOLE DERIVATIVES USEFUL AS KLK1 INHIBITORS VANTIA LIMITED (GB) 2011-05-05 WO disclosed