SCHEMBL1908467

SCHEMBL1908467

COc1ccncc1C#Cc1ccc(C2(N(C(=O)O)C(C)(C)C)CCC2)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.37
CYP2E1 P05181 1/20 0.37
CYP2A6 P11509 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2B6 P20813 1/20 0.37
CYP2C19 P33261 1/20 0.37
FFAR1 O14842 1/20 0.33
OPRM1 P35372 3/20 0.33
OPRL1 P41146 2/20 0.33
SLC22A12 Q96S37 2/20 0.32
GPBAR1 Q8TDU6 1/20 0.31
NR1H4 Q96RI1 1/20 0.31
HAO1 Q9UJM8 1/20 0.31
MMP12 P39900 1/20 0.30
PTGDR2 Q9Y5Y4 1/20 0.30
PTGES O14684 1/20 0.30
CA12 O43570 1/20 0.30
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30
CA9 Q16790 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2028947 0.78 GRM5 (0.37) FFAR1OPRM1OPRL1MMP12
SCHEMBL1900539 0.78 ACACB (0.30)
SCHEMBL1900135 0.78 CYP1A2 (0.39) CYP1A2CYP2E1CYP2A6CYP2C9CYP2B6
SCHEMBL1899248 0.77 FFAR1 (0.31) FFAR1OPRM1OPRL1PTGES
SCHEMBL14118801 0.76 AKT1 (0.36) CYP1A2CYP2E1CYP2A6CYP2C9CYP2B6
SCHEMBL1900125 0.75 CTSL (0.32) CYP2C9OPRM1OPRL1
SCHEMBL1352509 0.72 OPRL1 (0.39) CYP1A2CYP2C9OPRM1OPRL1
SCHEMBL2030849 0.70 OPRL1 (0.38) CYP1A2CYP2C9OPRM1OPRL1
SCHEMBL1902393 0.69 ROCK2 (0.38) FFAR1MMP12
SCHEMBL1352136 0.68 CCR2 (0.43) CYP1A2CYP2C9CYP2C19OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011055115-A1 AKT / PKB INHIBITORS ALMAC DISCOVERY LIMITED (GB) 2011-05-12 WO disclosed