SCHEMBL19085993

SCHEMBL19085993

CC[C@@H](NC(=O)c1ccc2[nH]ncc2c1)C(=O)N1CCc2sc(C(=O)Nc3cccc(C)c3C)cc2C1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
BTK Q06187 5/20 0.38
TDP1 Q9NUW8 1/20 0.37
LMNA P02545 2/20 0.37
MAPT P10636 2/20 0.37
KMT2A Q03164 2/20 0.37
ALDH1A1 P00352 1/20 0.37
RXFP1 Q9HBX9 1/20 0.36
ROCK2 O75116 2/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
PRMT5 O14744 2/20 0.36
WDR77 Q9BQA1 2/20 0.36
ROCK1 Q13464 1/20 0.36
DDR1 Q08345 2/20 0.36
MEN1 O00255 1/20 0.36
METTL3 Q86U44 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19086145 0.90 ROCK2 (0.36) BTKMAPTALDH1A1ROCK2PRMT5
SCHEMBL19085987 0.90 KDM1A (0.41) ALDH1A1ROCK2NPC1RAB9APRMT5
SCHEMBL19086004 0.89 PRMT5 (0.39) ROCK2NPC1RAB9APRMT5WDR77
SCHEMBL19086258 0.89 ROCK2 (0.34) BTKROCK2PRMT5WDR77ROCK1
SCHEMBL19085999 0.88 TRPV1 (0.41) KMT2AROCK2NPC1RAB9APRMT5
SCHEMBL19085981 0.88 TRPV1 (0.41) KMT2AROCK2NPC1RAB9APRMT5
SCHEMBL19086146 0.87 ROCK2 (0.35) BTKROCK2PRMT5WDR77ROCK1
SCHEMBL19085989 0.86 MAOB (0.41) ROCK2NPC1RAB9AROCK1
SCHEMBL19085978 0.86 ROCK2 (0.46) ROCK2NPC1RAB9APRMT5WDR77
SCHEMBL19086144 0.86 ROCK2 (0.35) MAPTROCK2PRMT5WDR77ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017114275-A1 COMPOUND FOR INHIBITING ROCK, PREPARATION METHOD AND USE OF SAME 成都先导药物开发有限公司 2017-07-06 WO disclosed