SCHEMBL19085998

SCHEMBL19085998

CC[C@@H](NC(=O)c1cc2cn[nH]c2cc1F)C(=O)N1CCc2sc(C(=O)Nc3ccccc3)cc2C1

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PRMT5 O14744 10/20 0.39
WDR77 Q9BQA1 10/20 0.39
KDM1A O60341 1/20 0.38
SMO Q99835 1/20 0.37
NPC1 O15118 1/20 0.36
HPGD P15428 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
JAK2 O60674 1/20 0.36
JAK1 P23458 1/20 0.36
TRPV1 Q8NER1 2/20 0.35
ACACB O00763 1/20 0.35
ACACA Q13085 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19085988 0.90 HCRTR2 (0.40) PRMT5WDR77SMONPC1HPGD
SCHEMBL19085981 0.90 TRPV1 (0.41) PRMT5WDR77SMONPC1RAB9A
SCHEMBL19085999 0.90 TRPV1 (0.41) PRMT5WDR77SMONPC1RAB9A
SCHEMBL19085977 0.86 NPC1 (0.45) PRMT5WDR77KDM1ANPC1RAB9A
SCHEMBL19085978 0.85 ROCK2 (0.46) PRMT5WDR77NPC1RAB9ATRPV1
SCHEMBL19085987 0.84 KDM1A (0.41) PRMT5WDR77KDM1ANPC1HPGD
SCHEMBL19085990 0.84 BRAF (0.40) PRMT5WDR77SMOHDAC6
SCHEMBL19085989 0.82 MAOB (0.41) NPC1RAB9A
SCHEMBL19086178 0.82 NPC1 (0.38) NPC1RAB9ATRPV1
SCHEMBL19086011 0.81 KDM1A (0.43) PRMT5WDR77KDM1ASMONPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017114275-A1 COMPOUND FOR INHIBITING ROCK, PREPARATION METHOD AND USE OF SAME 成都先导药物开发有限公司 2017-07-06 WO disclosed