SCHEMBL19085987

SCHEMBL19085987

CC[C@@H](NC(=O)c1ccc2[nH]ncc2c1)C(=O)N1CCc2sc(C(=O)Nc3ccccc3F)cc2C1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.41
ROCK2 O75116 7/20 0.39
ROCK1 Q13464 5/20 0.39
PRMT5 O14744 5/20 0.38
WDR77 Q9BQA1 5/20 0.38
HCRTR1 O43613 1/20 0.37
HCRTR2 O43614 1/20 0.37
CTNNB1 P35222 1/20 0.37
WNT3A P56704 1/20 0.37
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37
NPC1 O15118 1/20 0.37
TSHR P16473 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
GRIN2B Q13224 1/20 0.36
JAK2 O60674 1/20 0.36
JAK1 P23458 1/20 0.36
ANPEP P15144 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19085981 0.90 TRPV1 (0.41) ROCK2ROCK1PRMT5WDR77HCRTR2
SCHEMBL19085999 0.90 TRPV1 (0.41) ROCK2ROCK1PRMT5WDR77HCRTR2
SCHEMBL19085993 0.90 BTK (0.38) ROCK2ROCK1PRMT5WDR77ALDH1A1
SCHEMBL19086004 0.90 PRMT5 (0.39) KDM1AROCK2ROCK1PRMT5WDR77
SCHEMBL19086144 0.89 ROCK2 (0.35) KDM1AROCK2ROCK1PRMT5WDR77
SCHEMBL19085985 0.89 PRMT5 (0.40) ROCK2ROCK1PRMT5WDR77GRIN2B
SCHEMBL19085977 0.89 NPC1 (0.45) KDM1AROCK2ROCK1PRMT5WDR77
SCHEMBL19086145 0.88 ROCK2 (0.36) ROCK2ROCK1PRMT5WDR77ALDH1A1
SCHEMBL19085978 0.88 ROCK2 (0.46) ROCK2ROCK1PRMT5WDR77NPC1
SCHEMBL19085982 0.88 KDM4E (0.39) KDM1AROCK2ROCK1PRMT5WDR77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017114275-A1 COMPOUND FOR INHIBITING ROCK, PREPARATION METHOD AND USE OF SAME 成都先导药物开发有限公司 2017-07-06 WO disclosed