SCHEMBL19086177

SCHEMBL19086177

O=C(Nc1ccccc1)c1cc2c(s1)CCNC2

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PNMT P11086 2/20 0.58
ITGB3 P05106 5/20 0.52
ITGA2B P08514 5/20 0.52
MAPT P10636 8/20 0.51
NPC1 O15118 5/20 0.51
RAB9A P51151 5/20 0.51
ALDH1A1 P00352 5/20 0.51
SMN1; SMN2 Q16637 4/20 0.51
NFKB1 P19838 1/20 0.51
NFKB2 Q00653 1/20 0.51
RELA Q04206 1/20 0.51
LMNA P02545 4/20 0.46
KDM4E B2RXH2 4/20 0.46
HTT P42858 2/20 0.45
HPGD P15428 1/20 0.45
MEN1 O00255 1/20 0.45
GAA P10253 1/20 0.45
KMT2A Q03164 1/20 0.45
TPSAB1 Q15661 1/20 0.45
TPSD1 Q9BZJ3 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13822830 0.87 PNMT (0.59) PNMTITGB3ITGA2BMAPTNPC1
SCHEMBL8555210 0.83 ITGB3 (0.73) PNMTITGB3ITGA2BMAPTNPC1
SCHEMBL978035 0.83 PNMT (0.56) PNMTITGB3ITGA2BMAPTRAB9A
SCHEMBL28533972 0.79 PNMT (0.70) PNMTITGB3ITGA2BMAPTNPC1
SCHEMBL977949 0.78 PNMT (0.73) PNMTITGB3ITGA2BALDH1A1LMNA
Hydrochloric Acid SCHEMBL3441470 0.77 PNMT (0.71) PNMTITGB3ITGA2BALDH1A1LMNA
SCHEMBL6421837 0.74 PNMT (1.00) PNMTITGB3ITGA2BALDH1A1TPSAB1
SCHEMBL19086350 0.73 MAPT (0.48) MAPTNPC1RAB9AALDH1A1SMN1; SMN2
SCHEMBL977061 0.73 PNMT (0.70) PNMTITGB3ITGA2BMAPTNPC1
SCHEMBL14863153 0.73 PLAU (0.61) ITGB3ITGA2BNPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108239082-B Compound for inhibiting ROCK and application thereof 成都先导药物开发股份有限公司 2021-01-05 CN disclosed
WO-2017114275-A1 COMPOUND FOR INHIBITING ROCK, PREPARATION METHOD AND USE OF SAME 成都先导药物开发有限公司 2017-07-06 WO disclosed