SCHEMBL19086180

SCHEMBL19086180

CC[C@@H](NC(=O)c1ccc2[nH]ncc2c1)C(=O)N1CCc2sc(C(=O)N3CCOC(C)C3)cc2C1

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
METTL3 Q86U44 1/20 0.35
ACACB O00763 3/20 0.35
PIK3CA P42336 2/20 0.35
DDR1 Q08345 3/20 0.35
ALDH1A1 P00352 1/20 0.35
CYP1A2 P05177 1/20 0.35
HPGD P15428 1/20 0.35
CYP2C19 P33261 1/20 0.35
ROCK2 O75116 2/20 0.34
ROCK1 Q13464 2/20 0.34
PRMT5 O14744 3/20 0.34
WDR77 Q9BQA1 3/20 0.34
ACACA Q13085 2/20 0.33
AKT1 P31749 1/20 0.33
HDAC6 Q9UBN7 2/20 0.33
LIPC P11150 1/20 0.33
LIPG Q9Y5X9 1/20 0.33
PDE2A O00408 1/20 0.33
PDE3A Q14432 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19086182 0.91 SMO (0.40) METTL3ACACBPIK3CADDR1ROCK2
SCHEMBL19086147 0.84 ROCK2 (0.37) METTL3ACACBROCK2ROCK1PRMT5
SCHEMBL19086160 0.84 HDAC6 (0.38) METTL3ACACBROCK2ROCK1PRMT5
SCHEMBL19086049 0.84 ROCK2 (0.43) METTL3ROCK2ROCK1PRMT5WDR77
SCHEMBL19086054 0.84 ROCK2 (0.41) METTL3ACACBROCK2ROCK1PRMT5
SCHEMBL19086163 0.83 METTL3 (0.37) METTL3ACACBROCK2ROCK1PRMT5
SCHEMBL19086020 0.83 ROCK2 (0.44) ROCK2ROCK1PRMT5WDR77AKT1
SCHEMBL19086141 0.83 ROCK2 (0.44) ROCK2ROCK1PRMT5WDR77AKT1
SCHEMBL19086018 0.83 ROCK2 (0.44) METTL3ROCK2ROCK1AKT1HDAC6
SCHEMBL19086167 0.82 METTL3 (0.37) METTL3ROCK2HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017114275-A1 COMPOUND FOR INHIBITING ROCK, PREPARATION METHOD AND USE OF SAME 成都先导药物开发有限公司 2017-07-06 WO disclosed