SCHEMBL19086182

SCHEMBL19086182

CC[C@@H](NC(=O)c1ccc2[nH]ncc2c1)C(=O)N1CCc2sc(C(=O)N3CCOCC3)cc2C1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SMO Q99835 2/20 0.40
DDR1 Q08345 6/20 0.40
ROCK2 O75116 1/20 0.39
METTL3 Q86U44 1/20 0.37
ACACB O00763 3/20 0.37
ACACA Q13085 2/20 0.37
PIK3CA P42336 1/20 0.37
MAPK14 Q16539 1/20 0.37
BTK Q06187 1/20 0.36
NAMPT P43490 1/20 0.36
LRRK2 Q5S007 1/20 0.36
PRMT5 O14744 1/20 0.36
WDR77 Q9BQA1 1/20 0.36
PIN1 Q13526 1/20 0.36
KCNH2 Q12809 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19086180 0.91 METTL3 (0.35) DDR1ROCK2METTL3ACACBACACA
SCHEMBL19086049 0.88 ROCK2 (0.43) ROCK2METTL3MAPK14PRMT5WDR77
SCHEMBL19086147 0.87 ROCK2 (0.37) ROCK2METTL3ACACBACACAPRMT5
SCHEMBL19086160 0.87 HDAC6 (0.38) ROCK2METTL3ACACBACACANAMPT
SCHEMBL19086054 0.87 ROCK2 (0.41) ROCK2METTL3ACACBMAPK14PRMT5
SCHEMBL19086163 0.86 METTL3 (0.37) ROCK2METTL3ACACBACACAPRMT5
SCHEMBL19086018 0.86 ROCK2 (0.44) ROCK2METTL3MAPK14NAMPT
SCHEMBL19086167 0.85 METTL3 (0.37) ROCK2METTL3MAPK14BTKLRRK2
SCHEMBL19085999 0.85 TRPV1 (0.41) SMODDR1ROCK2PRMT5WDR77
SCHEMBL19086039 0.85 PRMT5 (0.39) ROCK2METTL3PRMT5WDR77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017114275-A1 COMPOUND FOR INHIBITING ROCK, PREPARATION METHOD AND USE OF SAME 成都先导药物开发有限公司 2017-07-06 WO disclosed