SCHEMBL19086216

SCHEMBL19086216

CC[C@@H](NC(=O)c1ccc(N)c(C=N)c1)C(=O)N1CCc2sc(C(=O)NC3CCNC3)cc2C1

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 3/20 0.35
KIFC1 Q9BW19 2/20 0.35
ACSS2 Q9NR19 1/20 0.34
PRMT5 O14744 8/20 0.33
WDR77 Q9BQA1 8/20 0.33
HCRTR2 O43614 2/20 0.33
KMT2A Q03164 1/20 0.33
KDM1A O60341 1/20 0.32
SUV39H1 O43463 1/20 0.32
PRMT1 Q99873 1/20 0.32
SMYD3 Q9H7B4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19086184 0.90 HDAC6 (0.37) HDAC6PRMT5WDR77HCRTR2KDM1A
SCHEMBL19086241 0.89 HDAC6 (0.36) HDAC6PRMT5WDR77KDM1A
SCHEMBL19086206 0.88 HDAC6 (0.38) HDAC6PRMT5WDR77HCRTR2KMT2A
SCHEMBL19086017 0.87 HDAC6 (0.36) HDAC6PRMT5WDR77KDM1A
SCHEMBL19086219 0.87 HDAC6 (0.36) HDAC6PRMT5WDR77KDM1ASMYD3
SCHEMBL19086335 0.85 HDAC6 (0.39) HDAC6PRMT5WDR77HCRTR2KMT2A
SCHEMBL19086201 0.83 PRMT5 (0.40) HDAC6PRMT5WDR77
SCHEMBL19086050 0.82 ROCK2 (0.41) HDAC6ACSS2
SCHEMBL19086194 0.81 PRMT5 (0.43) PRMT5WDR77HCRTR2KMT2A
SCHEMBL19086009 0.81 KMT2A (0.42) PRMT5WDR77HCRTR2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017114275-A1 COMPOUND FOR INHIBITING ROCK, PREPARATION METHOD AND USE OF SAME 成都先导药物开发有限公司 2017-07-06 WO disclosed