SCHEMBL19086230

SCHEMBL19086230

O=C(NCC(=O)N1CCc2sc(C(=O)Nc3cccc(Cl)c3)cc2C1)c1ccc2[nH]ncc2c1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAOB P27338 6/20 0.44
ROCK2 O75116 2/20 0.42
PRKD3 O94806 1/20 0.42
MAP4K4 O95819 1/20 0.42
RPS6KB1 P23443 1/20 0.42
CLK2 P49760 1/20 0.42
ROCK1 Q13464 1/20 0.42
DYRK1A Q13627 1/20 0.42
PRKG1 Q13976 1/20 0.42
PRKD2 Q9BZL6 1/20 0.42
CLK4 Q9HAZ1 1/20 0.42
SGK2 Q9HBY8 1/20 0.42
STK17A Q9UEE5 1/20 0.42
CCNE1 P24864 1/20 0.40
CDK2 P24941 1/20 0.40
MAOA P21397 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19086183 0.86 KDM1A (0.40) MAOBROCK2MAP4K4RPS6KB1CLK2
SCHEMBL19086026 0.85 METTL3 (0.44) MAOBROCK2ROCK1
SCHEMBL19085989 0.85 MAOB (0.41) MAOBROCK2PRKD3MAP4K4RPS6KB1
SCHEMBL19086995 0.81 ROCK2 (0.47) MAOBROCK2RPS6KB1ROCK1
SCHEMBL19086209 0.81 ROCK2 (0.43) MAOBROCK2ROCK1
SCHEMBL19086214 0.81 METTL3 (0.48) MAOBROCK2ROCK1
SCHEMBL19086190 0.80 ROCK2 (0.48) ROCK2PRKD3MAP4K4RPS6KB1ROCK1
SCHEMBL19086185 0.80 METTL3 (0.43) MAOBROCK2ROCK1
SCHEMBL19086208 0.80 KDM1A (0.44) MAOBMAOA
SCHEMBL19086217 0.79 ROCK2 (0.43) MAOBROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017114275-A1 COMPOUND FOR INHIBITING ROCK, PREPARATION METHOD AND USE OF SAME 成都先导药物开发有限公司 2017-07-06 WO disclosed