SCHEMBL19086208

SCHEMBL19086208

COc1ccc(F)cc1NC(=O)c1cc2c(s1)CCN(C(=O)CNC(=O)c1ccc3[nH]ncc3c1)C2

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 5/20 0.44
HDAC6 Q9UBN7 4/20 0.42
SMN1; SMN2 Q16637 4/20 0.41
KDM4E B2RXH2 2/20 0.41
RAB9A P51151 1/20 0.41
MAOB P27338 3/20 0.40
MAOA P21397 2/20 0.40
ALDH1A1 P00352 3/20 0.40
HTT P42858 2/20 0.40
HPGD P15428 2/20 0.40
MAPT P10636 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
GPR55 Q9Y2T6 2/20 0.38
LMNA P02545 1/20 0.38
CNR1 P21554 2/20 0.38
PRMT5 O14744 1/20 0.38
WDR77 Q9BQA1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19085982 0.86 KDM4E (0.39) KDM1ASMN1; SMN2KDM4ERAB9AMAOB
SCHEMBL19086223 0.85 METTL3 (0.43) KDM1AHDAC6KDM4EMAOBALDH1A1
SCHEMBL19086000 0.85 KDM4E (0.39) KDM1AHDAC6SMN1; SMN2KDM4ERAB9A
SCHEMBL19086026 0.84 METTL3 (0.44) KDM1AHDAC6SMN1; SMN2MAOBALDH1A1
SCHEMBL19086183 0.82 KDM1A (0.40) KDM1AHDAC6RAB9AMAOBL3MBTL1
SCHEMBL19086024 0.81 MAOB (0.43) KDM1AHDAC6KDM4EMAOBALDH1A1
SCHEMBL19086214 0.80 METTL3 (0.48) SMN1; SMN2MAOBALDH1A1HTTL3MBTL1
SCHEMBL19086230 0.80 MAOB (0.44) MAOBMAOA
SCHEMBL19086190 0.80 ROCK2 (0.48) KDM1AHDAC6
SCHEMBL19086259 0.79 METTL3 (0.42) KDM1AHDAC6SMN1; SMN2MAOBHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017114275-A1 COMPOUND FOR INHIBITING ROCK, PREPARATION METHOD AND USE OF SAME 成都先导药物开发有限公司 2017-07-06 WO disclosed