SCHEMBL19086249

SCHEMBL19086249

CCN1CCC(NC(=O)c2cc3c(s2)CCN(C(=O)CNC(=O)c2ccc4[nH]ncc4c2)C3)CC1

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 4/20 0.50
ROCK1 Q13464 2/20 0.50
MAPK14 Q16539 1/20 0.41
HDAC6 Q9UBN7 4/20 0.39
KDM1A O60341 3/20 0.39
METTL3 Q86U44 1/20 0.39
NAMPT P43490 1/20 0.38
DYRK1A Q13627 4/20 0.37
RPS6KB1 P23443 1/20 0.37
HTT P42858 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
PRMT5 O14744 1/20 0.37
WDR77 Q9BQA1 1/20 0.37
WNT1 P04628 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19086190 0.93 ROCK2 (0.48) ROCK2ROCK1MAPK14HDAC6KDM1A
SCHEMBL19086995 0.91 ROCK2 (0.47) ROCK2ROCK1MAPK14HDAC6KDM1A
SCHEMBL19086209 0.88 ROCK2 (0.43) ROCK2ROCK1MAPK14HDAC6KDM1A
SCHEMBL19086217 0.87 ROCK2 (0.43) ROCK2ROCK1MAPK14HDAC6KDM1A
SCHEMBL19086051 0.86 ROCK2 (0.48) ROCK2ROCK1MAPK14HDAC6DYRK1A
SCHEMBL19086026 0.86 METTL3 (0.44) ROCK2ROCK1HDAC6KDM1AMETTL3
SCHEMBL19086198 0.83 HDAC6 (0.38) ROCK2ROCK1HDAC6KDM1AMETTL3
SCHEMBL19086214 0.82 METTL3 (0.48) ROCK2ROCK1MAPK14METTL3HTT
SCHEMBL19086052 0.80 ROCK2 (0.46) ROCK2ROCK1MAPK14HDAC6DYRK1A
SCHEMBL19086020 0.79 ROCK2 (0.44) ROCK2ROCK1MAPK14HDAC6RPS6KB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017114275-A1 COMPOUND FOR INHIBITING ROCK, PREPARATION METHOD AND USE OF SAME 成都先导药物开发有限公司 2017-07-06 WO disclosed