SCHEMBL19086198

SCHEMBL19086198

CN1C=CC(NC(=O)c2cc3c(s2)CCN(C(=O)CNC(=O)c2ccc4[nH]ncc4c2)C3)N1

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 6/20 0.38
KDM1A O60341 4/20 0.38
METTL3 Q86U44 1/20 0.38
ROCK2 O75116 3/20 0.37
ROCK1 Q13464 1/20 0.37
ALDH1A1 P00352 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
PRMT5 O14744 6/20 0.36
WDR77 Q9BQA1 6/20 0.36
HTT P42858 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
MAOB P27338 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19086190 0.87 ROCK2 (0.48) HDAC6KDM1AMETTL3ROCK2ROCK1
SCHEMBL19086026 0.85 METTL3 (0.44) HDAC6KDM1AMETTL3ROCK2ROCK1
SCHEMBL19086209 0.84 ROCK2 (0.43) HDAC6KDM1AMETTL3ROCK2ROCK1
SCHEMBL19086995 0.84 ROCK2 (0.47) HDAC6KDM1AMETTL3ROCK2ROCK1
SCHEMBL19086249 0.83 ROCK2 (0.50) HDAC6KDM1AMETTL3ROCK2ROCK1
SCHEMBL19086217 0.82 ROCK2 (0.43) HDAC6KDM1AMETTL3ROCK2ROCK1
SCHEMBL19086214 0.81 METTL3 (0.48) METTL3ROCK2ROCK1ALDH1A1L3MBTL1
SCHEMBL19086185 0.79 METTL3 (0.43) HDAC6KDM1AMETTL3ROCK2ROCK1
SCHEMBL19086351 0.78 MAOB (0.44) HDAC6KDM1AMETTL3ROCK2PRMT5
SCHEMBL19086230 0.78 MAOB (0.44) ROCK2ROCK1MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017114275-A1 COMPOUND FOR INHIBITING ROCK, PREPARATION METHOD AND USE OF SAME 成都先导药物开发有限公司 2017-07-06 WO disclosed