SCHEMBL19086257

SCHEMBL19086257

CC[C@@H](NC(=O)c1ccc2[nH]ncc2c1)C(=O)N1CCc2sc(C(=O)Nc3cncc(C(F)(F)F)c3)cc2C1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PRMT5 O14744 2/20 0.38
WDR77 Q9BQA1 2/20 0.38
DDR2 Q16832 4/20 0.37
ABL1 P00519 2/20 0.37
ENPP2 Q13822 1/20 0.36
WNT1 P04628 1/20 0.36
TRPV1 Q8NER1 3/20 0.35
MAOB P27338 2/20 0.35
BCR P11274 1/20 0.35
HDAC6 Q9UBN7 1/20 0.34
MEN1 O00255 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
KMT2A Q03164 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
JAK3 P52333 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19086254 0.90 PRMT5 (0.40) PRMT5WDR77DDR2ENPP2MAOB
SCHEMBL19086256 0.89 NPC1 (0.41) PRMT5WDR77MAOBMEN1NPC1
SCHEMBL19085977 0.88 NPC1 (0.45) PRMT5WDR77MAOBHDAC6MEN1
SCHEMBL19085999 0.88 TRPV1 (0.41) PRMT5WDR77TRPV1MAOBNPC1
SCHEMBL19085981 0.88 TRPV1 (0.41) PRMT5WDR77TRPV1MAOBNPC1
SCHEMBL19085978 0.86 ROCK2 (0.46) PRMT5WDR77TRPV1MAOBNPC1
SCHEMBL19086178 0.85 NPC1 (0.38) TRPV1MAOBMEN1NPC1RAB9A
SCHEMBL19086255 0.85 MEN1 (0.39) TRPV1MAOBMEN1NPC1RAB9A
SCHEMBL19086167 0.85 METTL3 (0.37) TRPV1MAOBHDAC6MEN1NPC1
SCHEMBL19086169 0.84 METTL3 (0.37) DDR2ABL1TRPV1MAOBBCR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017114275-A1 COMPOUND FOR INHIBITING ROCK, PREPARATION METHOD AND USE OF SAME 成都先导药物开发有限公司 2017-07-06 WO disclosed