SCHEMBL19086320

SCHEMBL19086320

O=CN1CCc2sc(C(=O)NCc3ccccc3)cc2C1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.56
SMN1; SMN2 Q16637 3/20 0.56
MEN1 O00255 1/20 0.56
KMT2A Q03164 1/20 0.56
RXFP1 Q9HBX9 1/20 0.56
ALDH1A1 P00352 3/20 0.52
PRMT5 O14744 11/20 0.51
WDR77 Q9BQA1 11/20 0.51
LMNA P02545 2/20 0.46
NPC1 O15118 2/20 0.45
TP53 P04637 2/20 0.45
POLB P06746 2/20 0.45
HPGD P15428 2/20 0.45
RAB9A P51151 2/20 0.45
TSHR P16473 1/20 0.45
HTT P42858 1/20 0.45
MAPT P10636 1/20 0.43
HSD17B10 Q99714 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
ADORA1 P30542 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19087009 0.90 ALDH1A1 (0.49) KDM4ESMN1; SMN2MEN1KMT2ARXFP1
SCHEMBL19086028 0.79 ALDH1A1 (0.47) KDM4ESMN1; SMN2MEN1KMT2ARXFP1
SCHEMBL19086231 0.79 ALDH1A1 (0.56) KDM4ESMN1; SMN2MEN1KMT2AALDH1A1
SCHEMBL19087008 0.79 PRMT5 (0.41) KDM4ESMN1; SMN2MEN1KMT2ARXFP1
SCHEMBL19086022 0.74 RAB9A (0.56) KDM4ESMN1; SMN2MEN1KMT2ARXFP1
SCHEMBL19086996 0.70 NPC1 (0.45) SMN1; SMN2ALDH1A1PRMT5WDR77NPC1
SCHEMBL7797683 0.68 KMT2A (0.60) KDM4ESMN1; SMN2MEN1KMT2ARXFP1
SCHEMBL19086176 0.67 KDM1A (0.51) KDM4ESMN1; SMN2MEN1KMT2AALDH1A1
SCHEMBL1174282 0.66 HDAC6 (0.54) KDM4ESMN1; SMN2MEN1KMT2AALDH1A1
SCHEMBL21428365 0.66 PDE4D (0.44) SMN1; SMN2NPC1RAB9ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017114275-A1 COMPOUND FOR INHIBITING ROCK, PREPARATION METHOD AND USE OF SAME 成都先导药物开发有限公司 2017-07-06 WO disclosed