SCHEMBL19086351

SCHEMBL19086351

Cc1cc(CNC(=O)c2cc3c(s2)CCN(C(=O)CNC(=O)c2ccc4[nH]ncc4c2)C3)ccn1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAOB P27338 1/20 0.44
METTL3 Q86U44 1/20 0.43
ROCK2 O75116 6/20 0.42
NAMPT P43490 2/20 0.39
TLR9 Q9NR96 1/20 0.37
TLR8 Q9NR97 1/20 0.37
TLR7 Q9NYK1 1/20 0.37
PRMT5 O14744 3/20 0.37
WDR77 Q9BQA1 3/20 0.37
KDM1A O60341 3/20 0.37
HDAC6 Q9UBN7 3/20 0.37
HTT P42858 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
SLC8A1 P32418 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19086349 0.87 MAOB (0.40) MAOBMETTL3ROCK2NAMPTPRMT5
SCHEMBL19086026 0.85 METTL3 (0.44) MAOBMETTL3ROCK2PRMT5WDR77
SCHEMBL19086024 0.85 MAOB (0.43) MAOBMETTL3ROCK2NAMPTPRMT5
SCHEMBL19086259 0.84 METTL3 (0.42) MAOBMETTL3ROCK2NAMPTPRMT5
SCHEMBL19086223 0.83 METTL3 (0.43) MAOBMETTL3ROCK2NAMPTPRMT5
SCHEMBL19086214 0.83 METTL3 (0.48) MAOBMETTL3ROCK2HTTSMN1; SMN2
SCHEMBL19086183 0.82 KDM1A (0.40) MAOBMETTL3ROCK2KDM1AHDAC6
SCHEMBL19086190 0.81 ROCK2 (0.48) METTL3ROCK2KDM1AHDAC6
SCHEMBL19086209 0.80 ROCK2 (0.43) MAOBMETTL3ROCK2NAMPTPRMT5
SCHEMBL19086995 0.80 ROCK2 (0.47) MAOBMETTL3ROCK2PRMT5WDR77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017114275-A1 COMPOUND FOR INHIBITING ROCK, PREPARATION METHOD AND USE OF SAME 成都先导药物开发有限公司 2017-07-06 WO disclosed