SCHEMBL19086259

SCHEMBL19086259

Cc1cc(F)ncc1CNC(=O)c1cc2c(s1)CCN(C(=O)CNC(=O)c1ccc3[nH]ncc3c1)C2

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
METTL3 Q86U44 1/20 0.42
KDM1A O60341 5/20 0.39
HDAC6 Q9UBN7 5/20 0.39
MAOB P27338 1/20 0.38
NAMPT P43490 2/20 0.37
PRMT5 O14744 4/20 0.36
WDR77 Q9BQA1 4/20 0.36
HTT P42858 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
ROCK2 O75116 1/20 0.35
ENPP2 Q13822 1/20 0.35
DDR1 Q08345 1/20 0.35
BTK Q06187 1/20 0.35
KLKB1 P03952 1/20 0.35
MAP4K1 Q92918 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19086223 0.89 METTL3 (0.43) METTL3KDM1AHDAC6MAOBNAMPT
SCHEMBL19086260 0.87 METTL3 (0.38) METTL3MAOBNAMPTPRMT5WDR77
SCHEMBL19086351 0.84 MAOB (0.44) METTL3KDM1AHDAC6MAOBNAMPT
SCHEMBL19086026 0.84 METTL3 (0.44) METTL3KDM1AHDAC6MAOBPRMT5
SCHEMBL19086024 0.83 MAOB (0.43) METTL3KDM1AHDAC6MAOBNAMPT
SCHEMBL19086183 0.83 KDM1A (0.40) METTL3KDM1AHDAC6MAOBROCK2
SCHEMBL19086214 0.82 METTL3 (0.48) METTL3MAOBHTTSMN1; SMN2ROCK2
SCHEMBL19086190 0.80 ROCK2 (0.48) METTL3KDM1AHDAC6ROCK2
SCHEMBL19086208 0.79 KDM1A (0.44) KDM1AHDAC6MAOBPRMT5WDR77
SCHEMBL19086209 0.79 ROCK2 (0.43) METTL3KDM1AHDAC6MAOBNAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017114275-A1 COMPOUND FOR INHIBITING ROCK, PREPARATION METHOD AND USE OF SAME 成都先导药物开发有限公司 2017-07-06 WO disclosed