(R,S)-Ampa

(R,S)-Ampa

SCHEMBL19086372

Cc1onc(O)c1CC(N)C(=O)O.N[C@@H](CCC(=O)O)C(=O)O

nearest known ligand 0.58

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIA1 P42261 6/20 0.58
GRIA3 P42263 6/20 0.58
GRIA2 P42262 5/20 0.55
GRIA4 P48058 5/20 0.55
GRIK1 P39086 3/20 0.49
GRIK5 Q16478 3/20 0.49
CYP1A2 P05177 3/20 0.49
GRM6 O15303 3/20 0.49
GRIK2 Q13002 2/20 0.49
GRIK3 Q13003 2/20 0.49
GRM8 O00222 1/20 0.49
GRIN2D O15399 1/20 0.49
GRIN3B O60391 1/20 0.49
GSR P00390 1/20 0.49
GRM5 P41594 1/20 0.49
SLC1A3 P43003 1/20 0.49
SLC1A2 P43004 1/20 0.49
SLC1A1 P43005 1/20 0.49
GRIN1 Q05586 1/20 0.49
GRIN2A Q12879 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
(R,S)-Ampa SCHEMBL23242452 1.00 GRIA1 (0.58) GRIA1GRIA3GRIA2GRIA4GRIK1
(R,S)-Ampa SCHEMBL68799 0.90 GRIA1 (0.69) GRIA1GRIA3GRIA2GRIA4GRIK1
(R,S)-Ampa SCHEMBL2458874 0.90 GRIA1 (0.69) GRIA1GRIA3GRIA2GRIA4GRIK1
(S)-Ampa SCHEMBL667915 0.90 GRIA1 (0.69) GRIA1GRIA3GRIA2GRIA4GRIK1
(R,S)-Ampa SCHEMBL7200262 0.89 GRIA1 (0.68) GRIA1GRIA3GRIA2GRIA4GRIK1
(R,S)-Ampa SCHEMBL7200264 0.89 GRIA1 (0.68) GRIA1GRIA3GRIA2GRIA4GRIK1
(R,S)-Ampa SCHEMBL6553747 0.87 GRIA1 (0.56) GRIA1GRIA3GRIA2GRIA4GRIK1
SCHEMBL3731488 0.81 GRIA1 (0.54) GRIA1GRIA3GRIA2GRIA4GRIK1
SCHEMBL12506417 0.81 GRIA1 (0.54) GRIA1GRIA3GRIA2GRIA4GRIK1
(S)-Ampa SCHEMBL28091565 0.80 GRIA1 (0.53) GRIA1GRIA3GRIA2GRIA4GRIK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3190181-B1 CORNEAL ENDOTHELIAL CELL MARKER UNIV OSAKA (JP) 2020-06-17 EP disclosed
US-20170253855-A1 CORNEAL ENDOTHELIAL CELL MARKER OSAKA UNIVERSITY (JP) 2017-09-07 US disclosed
EP-3190181-A1 CORNEAL ENDOTHELIAL CELL MARKER Osaka University (JP) 2017-07-12 EP disclosed