(S)-Ampa

(S)-Ampa

SCHEMBL28091565

CN[C@H](CC(=O)O)C(=O)O.Cc1onc(O)c1C[C@H](N)C(=O)O

nearest known ligand 0.53

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIA1 P42261 5/20 0.53
GRIA3 P42263 5/20 0.53
GRIA2 P42262 4/20 0.51
GRIA4 P48058 4/20 0.51
MAPT P10636 2/20 0.39
GRIK1 P39086 2/20 0.39
GRIK5 Q16478 2/20 0.39
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
TSHR P16473 1/20 0.39
CYP2C19 P33261 1/20 0.39
KMT2A Q03164 1/20 0.39
GRIK2 Q13002 1/20 0.39
GRIK3 Q13003 1/20 0.39
GRIK4 Q16099 1/20 0.39
MAPK1 P28482 1/20 0.39
BLM P54132 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
(R,S)-Ampa SCHEMBL2458874 0.85 GRIA1 (0.69) GRIA1GRIA3GRIA2GRIA4MAPT
(S)-Ampa SCHEMBL667915 0.85 GRIA1 (0.69) GRIA1GRIA3GRIA2GRIA4MAPT
(R,S)-Ampa SCHEMBL68799 0.85 GRIA1 (0.69) GRIA1GRIA3GRIA2GRIA4MAPT
(R,S)-Ampa SCHEMBL7200262 0.84 GRIA1 (0.68) GRIA1GRIA3GRIA2GRIA4MAPT
(R,S)-Ampa SCHEMBL7200264 0.84 GRIA1 (0.68) GRIA1GRIA3GRIA2GRIA4MAPT
(R,S)-Ampa SCHEMBL23242452 0.80 GRIA1 (0.58) GRIA1GRIA3GRIA2GRIA4MAPT
(R,S)-Ampa SCHEMBL19086372 0.80 GRIA1 (0.58) GRIA1GRIA3GRIA2GRIA4MAPT
(R,S)-Ampa SCHEMBL6553747 0.78 GRIA1 (0.56) GRIA1GRIA3GRIA2GRIA4MAPT
SCHEMBL28471680 0.77 GRIA1 (0.47) GRIA1GRIA3GRIA2GRIA4MAPT
SCHEMBL24115240 0.74 GRIA1 (0.37) GRIA1GRIA3GRIA2GRIA4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105873570-A Sustained release depot formulations of therapeutic proteins and uses thereof 奇尼塔有限责任公司 2016-08-17 CN disclosed