SCHEMBL19086409

SCHEMBL19086409

CN(CCCOc1ccc(I)cc1)C(=O)O

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PDE1A P54750 7/20 0.50
PDE1B Q01064 7/20 0.50
PDE1C Q14123 7/20 0.50
KDM4E B2RXH2 3/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
ALDH1A1 P00352 2/20 0.49
LTA4H P09960 1/20 0.47
HRH3 Q9Y5N1 1/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
LSS P48449 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21114008 0.94 KDM4E (0.55) PDE1APDE1BPDE1CKDM4ESMN1; SMN2
SCHEMBL19553110 0.82 KDM4E (0.56) KDM4ESMN1; SMN2ALDH1A1KMT2A
SCHEMBL27164572 0.81 SMN1; SMN2 (0.53) KDM4ESMN1; SMN2ALDH1A1LTA4HHRH3
SCHEMBL17572343 0.81 PDK2 (0.47) PDE1APDE1BPDE1CKDM4ESMN1; SMN2
SCHEMBL10877728 0.80 LTA4H (0.69) KDM4ESMN1; SMN2ALDH1A1LTA4H
SCHEMBL5637895 0.79 KDM4E (0.69) PDE1APDE1BPDE1CKDM4ESMN1; SMN2
SCHEMBL2476605 0.77 KDM4E (0.49) KDM4ESMN1; SMN2ALDH1A1LTA4HMEN1
SCHEMBL21595690 0.77 DRD2 (0.60) KDM4ESMN1; SMN2MEN1KMT2A
SCHEMBL7994823 0.76 LTA4H (0.56) KDM4ESMN1; SMN2ALDH1A1LTA4HMEN1
SCHEMBL21163143 0.76 PDK2 (0.45) PDE1APDE1BPDE1CKDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3190111-B1 PYRAZOLO[3,4-C]PYRIDINE DERIVATIVES CSPC ZHONGQI PHARMACEUTICAL TECH SHIJIAZHUANG CO LTD (CN) 2020-05-06 EP disclosed
US-9975893-B2 Pyrazolo[3,4-c]pyridine derivatives CSPC ZHONGQI PHARMACEUTICAL TECHNOLOGY (SHIJIAZHUANG) CO., LTD. (CN) 2018-05-22 US disclosed
US-20170291896-A1 PYRAZOLO[3,4-C]PYRIDINE DERIVATIVES CSPC ZHONGQI PHARMACEUTICAL TECHNOLOGY (SHIJIAZHUANG) CO., LTD. (CN) 2017-10-12 US disclosed
EP-3190111-A1 PYRAZOLO[3,4-C]PYRIDINE DERIVATIVES CSPC Zhongqi Pharmaceutical Technology (Shijiazhuang) Co., Ltd. (CN) 2017-07-12 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170291896-A1 PYRAZOLO[3,4-C]PYRIDINE DERIVATIVES F11, TFPI, F2 PDE1A 529/4885PDE1B 705/4885PDE1C 872/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.