SCHEMBL19088802

SCHEMBL19088802

CC(C)(C)OC(=O)N1CCC(OC(=O)Nc2ccsc2-c2cccc(F)c2)CC1

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 1/20 0.46
GPR119 Q8TDV5 3/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC2 Q92769 1/20 0.43
TP53 P04637 2/20 0.42
CHRM3 P20309 7/20 0.41
CHRM2 P08172 1/20 0.41
CHRM1 P11229 1/20 0.41
PTPN2 P17706 1/20 0.41
PTPN1 P18031 1/20 0.41
PTPN6 P29350 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19088797 0.90 PTPN2 (0.47) GPR119HDAC1HDAC2PTPN2PTPN1
SCHEMBL19088794 0.89 STS (0.47) GPR119TP53CHRM3CHRM2CHRM1
SCHEMBL19066214 0.89 CHRM3 (0.48) GPR119CHRM3PTPN2PTPN1PTPN6
SCHEMBL19088791 0.84 CHRM3 (0.45) GPR119CHRM3
SCHEMBL19088795 0.80 CHRM3 (0.53) HDAC1HDAC2CHRM3CHRM2CHRM1
SCHEMBL19088803 0.79 PTPN2 (0.46) GPR119PTPN2PTPN1PTPN6
SCHEMBL4983940 0.78 GPR119 (0.48) HPGDSGPR119HDAC1HDAC2CHRM3
SCHEMBL14228062 0.78 HPGDS (0.45) HPGDSGPR119HDAC1HDAC2CHRM3
SCHEMBL19066183 0.77 CHRM3 (0.50) GPR119CHRM3PTPN2PTPN1PTPN6
SCHEMBL24906656 0.75 CHRM3 (0.70) CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107849035-B Phenyl heterocyclic derivative and application thereof in medicine 四川海思科制药有限公司 2021-12-10 CN disclosed
CN-107849035-A Phenyl heterocyclic derivative and application thereof in medicine 四川海思科制药有限公司 2018-03-27 CN disclosed
WO-2017114377-A1 BENZYL HETEROCYCLIC COMPOUND DERIVATIVE AND PHARMACEUTICAL APPLICATION THEREOF 四川海思科制药有限公司 2017-07-06 WO disclosed