SCHEMBL19089701

SCHEMBL19089701

C=N/C(C=O)=C\C=C(/C)c1cccc(C(F)(F)F)c1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
ALDH1A1 P00352 2/20 0.43
NPSR1 Q6W5P4 1/20 0.42
GAA P10253 2/20 0.40
SRD5A2 P31213 1/20 0.40
MAOB P27338 1/20 0.40
POLB P06746 1/20 0.40
HDAC3 O15379 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC2 Q92769 1/20 0.40
P2RX1 P51575 1/20 0.39
LMNA P02545 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28108408 0.81 CES2 (0.56) CES2MEN1KMT2AALDH1A1NPSR1
SCHEMBL19089736 0.79 TP53 (0.49) MEN1KMT2AALDH1A1NPSR1GAA
SCHEMBL9111870 0.75 CES2 (0.55) CES2MEN1KMT2AALDH1A1NPSR1
SCHEMBL9111866 0.75 CES2 (0.55) CES2MEN1KMT2AALDH1A1NPSR1
SCHEMBL19592309 0.74 CES2 (0.58) CES2MEN1KMT2AALDH1A1NPSR1
SCHEMBL20806278 0.73 CES2 (0.56) CES2MEN1KMT2AALDH1A1NPSR1
SCHEMBL6703582 0.71 NR4A1 (0.66) CES2MEN1KMT2AALDH1A1NPSR1
SCHEMBL6703585 0.71 NR4A1 (0.66) CES2MEN1KMT2AALDH1A1NPSR1
SCHEMBL7961946 0.70 CES2 (0.57) CES2MEN1KMT2AALDH1A1NPSR1
SCHEMBL7961951 0.70 CES2 (0.57) CES2MEN1KMT2AALDH1A1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10018619-B2 Compounds and method of identifying, synthesizing, optimizing and profiling protein modulators HMI Medical Innovations, LLC (US) 2018-07-10 US disclosed
US-20170191986-A1 Compounds and Method of Identifying, Synthesizing, Optimizing and Profiling Protein Modulators HMI Medical Innovations, LLC 2017-07-06 US disclosed