SCHEMBL19089786

SCHEMBL19089786

O=C(NNc1ccc2cc(-c3ccc(C(=O)NNc4ccc5ccccc5n4)c(O)c3)ccc2n1)c1ccccn1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM5A P29375 1/20 0.45
KDM4E B2RXH2 5/20 0.43
NPC1 O15118 4/20 0.43
RAB9A P51151 3/20 0.43
ALDH1A1 P00352 1/20 0.43
TP53 P04637 1/20 0.43
TSHR P16473 1/20 0.43
NFKB1 P19838 1/20 0.43
NFKB2 Q00653 1/20 0.43
RELA Q04206 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
GAA P10253 4/20 0.42
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
MAPT P10636 2/20 0.42
TDP1 Q9NUW8 2/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
HTT P42858 2/20 0.42
HDAC1 Q13547 1/20 0.42
POLB P06746 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4411512 0.84 KDM5A (0.60) KDM5AKDM4ENPC1RAB9AALDH1A1
SCHEMBL4414176 0.75 KDM4E (0.59) KDM4ENPC1RAB9AALDH1A1TP53
SCHEMBL6451494 0.67 KDM4E (0.58) KDM4ENPC1RAB9AALDH1A1SMN1; SMN2
SCHEMBL4407887 0.67 SORT1 (0.49) KDM4ENPC1RAB9AALDH1A1SMN1; SMN2
SCHEMBL21711110 0.67 NPC1 (0.49) KDM4ENPC1RAB9AALDH1A1TP53
SCHEMBL23388826 0.67 SMN1; SMN2 (0.61) KDM5AKDM4ENPC1RAB9AALDH1A1
SCHEMBL29995352 0.67 SMN1; SMN2 (0.61) KDM5AKDM4ENPC1RAB9AALDH1A1
SCHEMBL4542670 0.64 KDM4E (0.54) KDM4ENPC1RAB9AALDH1A1SMN1; SMN2
SCHEMBL1147702 0.63 KDM4E (0.73) KDM5AKDM4ENPC1RAB9AALDH1A1
SCHEMBL10062372 0.63 KDM5A (1.00) KDM5AKDM4ENPC1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11714080-B2 Compounds and methods of identifying, synthesizing, optimizing and profiling protein modulators HMI Medical Innovations, LLC (US) 2023-08-01 US disclosed
US-20210215671-A1 COMPOUNDS AND METHODS OF IDENTIFYING, SYNTHESIZING, OPTIMIZING AND PROFILING PROTEIN MODULATORS HMI Medical Innovations, LLC 2021-07-15 US disclosed
US-10018619-B2 Compounds and method of identifying, synthesizing, optimizing and profiling protein modulators HMI Medical Innovations, LLC (US) 2018-07-10 US disclosed
US-20170191986-A1 Compounds and Method of Identifying, Synthesizing, Optimizing and Profiling Protein Modulators HMI Medical Innovations, LLC 2017-07-06 US disclosed