SCHEMBL19112893

SCHEMBL19112893

CC(C)(C)O[C@H](O)N1C[C@H](O)C[C@H]1C(=O)N1CCC(CC(=O)Nc2cc(C(F)(F)F)cc(C(F)(F)F)c2)CC1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 4/20 0.40
CXCR3 P49682 2/20 0.40
ALDH1A1 P00352 2/20 0.35
NAMPT P43490 1/20 0.35
HCRTR1 O43613 1/20 0.35
HCRTR2 O43614 1/20 0.35
RHOC P08134 3/20 0.34
RHOA P61586 3/20 0.34
KCNH2 Q12809 1/20 0.34
CACNA1I Q9P0X4 1/20 0.34
USP30 Q70CQ3 1/20 0.34
LMNA P02545 1/20 0.33
STS P08842 1/20 0.33
GAA P10253 1/20 0.33
TACR1 P25103 1/20 0.33
ACP1 P24666 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4276573 0.83 CYP1A2 (0.43) EPHX2CXCR3ALDH1A1RHOCRHOA
SCHEMBL4276575 0.83 CYP1A2 (0.43) EPHX2CXCR3ALDH1A1RHOCRHOA
SCHEMBL8374022 0.77 CYP1A2 (0.40) EPHX2CXCR3STSTACR1
SCHEMBL6863335 0.75 STS (0.56) EPHX2CXCR3STSTACR1
SCHEMBL4272965 0.74 HSD17B10 (0.52) EPHX2CXCR3ALDH1A1HCRTR1HCRTR2
SCHEMBL4272968 0.74 HSD17B10 (0.52) EPHX2CXCR3ALDH1A1HCRTR1HCRTR2
SCHEMBL4276665 0.74 HSD17B10 (0.52) EPHX2CXCR3ALDH1A1HCRTR1HCRTR2
SCHEMBL4278127 0.74 CXCR3 (0.56) EPHX2CXCR3ALDH1A1NAMPTRHOC
SCHEMBL22019439 0.74 CXCR3 (0.46) EPHX2CXCR3ALDH1A1NAMPTHCRTR1
SCHEMBL1445327 0.74 LMNA (0.52) EPHX2CXCR3ALDH1A1NAMPTRHOC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3189839-A1 N-PIPERIDINYL ACETAMIDE DERIVATIVES AS CALCIUM CHANNEL BLOCKERS Taro Pharmaceuticals Inc. (CA) 2017-07-12 EP disclosed