SCHEMBL22019439

SCHEMBL22019439

CN1CCCC1C(=O)N1CCC(CC(=O)Nc2cc(C(F)(F)F)cc(C(F)(F)F)c2)CC1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CXCR3 P49682 3/20 0.46
EPHX2 P34913 4/20 0.46
HCRTR1 O43613 1/20 0.45
HCRTR2 O43614 1/20 0.45
NAMPT P43490 1/20 0.43
WNT3 P56703 1/20 0.42
SFRP1 Q8N474 1/20 0.42
KCNH2 Q12809 1/20 0.42
CACNA1I Q9P0X4 1/20 0.42
GAA P10253 1/20 0.41
LMNA P02545 1/20 0.41
RHOC P08134 3/20 0.41
RHOA P61586 3/20 0.41
ACP1 P24666 1/20 0.40
ALDH1A1 P00352 1/20 0.40
THRB P10828 1/20 0.39
CTSS P25774 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12004594 0.91 CXCR3 (0.44) CXCR3EPHX2HCRTR1HCRTR2NAMPT
SCHEMBL12004663 0.88 RHOC (0.44) CXCR3HCRTR1HCRTR2NAMPTWNT3
SCHEMBL6863162 0.87 CXCR3 (0.42) CXCR3EPHX2HCRTR1HCRTR2NAMPT
SCHEMBL1444264 0.84 EPHX2 (0.49) CXCR3EPHX2NAMPTKCNH2RHOC
SCHEMBL4272965 0.83 HSD17B10 (0.52) CXCR3EPHX2HCRTR1HCRTR2WNT3
SCHEMBL4272968 0.83 HSD17B10 (0.52) CXCR3EPHX2HCRTR1HCRTR2WNT3
SCHEMBL4276665 0.83 HSD17B10 (0.52) CXCR3EPHX2HCRTR1HCRTR2WNT3
SCHEMBL4274713 0.81 HSD17B10 (0.48) CXCR3EPHX2HCRTR1HCRTR2NAMPT
SCHEMBL1445327 0.81 LMNA (0.52) CXCR3EPHX2NAMPTGAALMNA
SCHEMBL12005602 0.79 RHOA (0.45) CXCR3EPHX2RHOCRHOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3189839-B1 N-PIPERIDINYL ACETAMIDE DERIVATIVES AS CALCIUM CHANNEL BLOCKERS PRAXIS PREC MEDICINES INC (US) 2020-05-20 EP disclosed